VR1 Activators
Items 11 to 18 of 18 total
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| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
Arvanil | 128007-31-8 | sc-202065 | 5 mg | $150.00 | 1 | |
Arvanil is a synthetic compound that acts as a potent agonist of the TRPV1 receptor, characterized by its unique ability to form stable interactions through van der Waals forces and ionic bonds. Its distinct molecular structure facilitates enhanced receptor affinity, leading to efficient activation. The compound's kinetic profile reveals rapid onset of action, influencing downstream signaling pathways and calcium influx, thereby modulating sensory perception and thermal nociception. | ||||||
PPAHV | 175796-50-6 | sc-202296 | 1 mg | $135.00 | ||
PPAHV is a specialized acid halide that exhibits remarkable reactivity due to its electrophilic nature, allowing it to readily engage in nucleophilic acyl substitution reactions. Its unique steric configuration enhances selectivity in reactions with amines and alcohols, promoting the formation of stable intermediates. The compound's ability to participate in diverse reaction pathways, including acylation and esterification, showcases its versatility in organic synthesis, while its physical properties contribute to its solubility and reactivity profile. | ||||||
6′-Iodoresiniferatoxin | 335151-55-8 | sc-202025 | 1 mg | $472.00 | ||
6′-Iodoresiniferatoxin is a potent modulator of the VR1 receptor, known for its unique ability to induce calcium influx in sensory neurons. Its iodine substituent enhances hydrophobic interactions, facilitating binding to the receptor's transmembrane domain. This compound exhibits distinct kinetics, with rapid activation and prolonged receptor desensitization, influencing pain signaling pathways. Its structural features allow for selective engagement with specific ion channels, highlighting its role in sensory transduction. | ||||||
Anandamide | 94421-68-8 | sc-396321 sc-396321A sc-396321B sc-396321C | 5 mg 25 mg 500 mg 1 g | $81.00 $219.00 $4068.00 $7813.00 | 2 | |
Anandamide is an endogenous cannabinoid that interacts with the VR1 receptor, exhibiting a unique affinity for lipid bilayers due to its hydrophobic tail. This interaction promotes conformational changes in the receptor, leading to calcium ion influx and subsequent neuronal signaling. Anandamide's rapid degradation by fatty acid amide hydrolase introduces a dynamic aspect to its action, influencing the temporal response in sensory pathways. Its dual role as a signaling molecule and modulator of receptor activity underscores its complexity in neurobiology. | ||||||
JYL-79 | sc-221785 sc-221785A | 1 mg 5 mg | $41.00 $218.00 | |||
JYL-79 is a potent acid halide that selectively engages with the VR1 receptor, facilitating unique hydrogen bonding interactions that enhance receptor activation. Its structural rigidity allows for precise orientation within the binding site, promoting efficient signal transduction. The compound exhibits rapid hydrolysis, generating reactive intermediates that can modulate downstream signaling pathways. This dynamic behavior contributes to its distinctive role in sensory perception and cellular communication. | ||||||
Probenecid-d14 | sc-219644 | 1 mg | $278.00 | |||
Probenecid-d14 is a specialized compound that interacts with the VR1 receptor through unique hydrophobic and electrostatic interactions, enhancing receptor sensitivity. Its isotopic labeling allows for precise tracking in metabolic studies, revealing insights into receptor dynamics. The compound's stability under physiological conditions enables prolonged engagement with the receptor, influencing downstream signaling cascades. This behavior underscores its role in modulating sensory pathways and cellular responses. | ||||||
JYL-1511 | 623166-14-3 | sc-202677 sc-202677A | 1 mg 5 mg | $200.00 $400.00 | ||
JYL-1511 is a distinctive acid halide that exhibits selective reactivity with nucleophiles, facilitating unique acylation processes. Its structure promotes rapid formation of stable intermediates, enhancing reaction kinetics in synthetic pathways. The compound's ability to form strong hydrogen bonds with surrounding molecules influences solubility and reactivity profiles, making it a versatile agent in various chemical transformations. Its distinct electronic properties contribute to its behavior in complex reaction environments. | ||||||
JYL-273 | 289902-71-2 | sc-202678 sc-202678A | 1 mg 5 mg | $48.00 $192.00 | ||
JYL-273 is a specialized acid halide characterized by its unique electrophilic nature, which allows for efficient acyl transfer reactions. The compound's steric configuration enhances its interaction with various nucleophiles, leading to the formation of diverse acyl derivatives. Its reactivity is influenced by the presence of electron-withdrawing groups, which stabilize transition states and accelerate reaction rates. Additionally, JYL-273 exhibits notable solvation effects, impacting its behavior in different solvent systems. | ||||||