Histamine H1 Receptor Inhibitors

Santa Cruz Biotechnology now offers a broad range of Histamine H1 Receptor Inhibitors. Histamine is an inflammatory mediator that is ubiquitously expressed and has a broad range of pharmacologic effects. The effects of histamine are mediated by a family of G protein-coupled receptors, the Histamine H1, H2, H3 and H4 Receptors. Histamine H1 Receptor Inhibitors offered by Santa Cruz inhibit Histamine H1 Receptor and, in some cases, other inflammation and immune response related proteins. View detailed Histamine H1 Receptor Inhibitor specifications, including Histamine H1 Receptor Inhibitor CAS number, molecular weight, molecular formula and chemical structure, by clicking on the product name.

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PRODUCT NAME/Application CAS Catalog # QUANTITY Price Citations RATING
Ketotifen fumarate
A histamine H1 antagonist and mast cell growth inhibitor
34580-14-8 sc-201094
sc-201094A
1 g
100 mg
$62.00
$39.00
3
(1)
Loratadine
Loratadine is a peripheral histamine H1 receptor agonist
79794-75-5 sc-203117
sc-203117A
10 mg
50 mg
$105.00
$446.00
1
(1)
Chlorpromazine, Hydrochloride
Chlorpromazine, Hydrochloride is an inhibitor of PDE, D2DR, NOS1, and PLA2
69-09-0 sc-202537
sc-202537A
sc-202537B
sc-202537C
sc-202537D
500 mg
5 g
25 g
100 g
250 g
$32.00
$48.00
$140.00
$480.00
$1,060.00
5
(1)
Terfenadine
Terfenadine is a histamine H1-receptor antagonist, which blocks HERG and KIR6 channels
50679-08-8 sc-208421A
sc-208421B
sc-208421
500 mg
1 g
5 g
$37.00
$64.00
$105.00
0
(1)
Astemizole
Astemizole is a potent and selective H1-receptor antagonist that displays antihistamine and antimalarial activity
68844-77-9 sc-201088
sc-201088A
10 mg
50 mg
$69.00
$275.00
2
(1)
Methapyrilene HCl
Methapyrilene HCl is a specialty product for proteomics research
135-23-9 sc-257708
1 g
$94.00
0
(0)
Diphenhydramine hydrochloride
Diphenhydramine hydrochloride is a histamine H1-receptor antagonist
147-24-0 sc-204729
sc-204729A
sc-204729B
10 g
25 g
100 g
$50.00
$80.00
$120.00
2
(1)
Meclizine Dihydrochloride
Meclizine Dihydrochloride is a histamine H1 receptor antagonist and PXR (pregnane X receptor) agonist
1104-22-9 sc-211779A
sc-211779
5 g
10 g
$20.00
$40.00
3
(1)
(S)-(+)-Dimethindene maleate
(S)-(+)-Dimethindene maleate is a subtype-selective mAChR M2 antagonist and histamine H1 receptor antagonist
121367-05-3 sc-361329
sc-361329A
10 mg
50 mg
$170.00
$700.00
0
(0)
Mepyramine maleate
Mepyramine maleate is a histamine H1 receptor antagonist
59-33-6 sc-203629
sc-203629A
100 mg
1 g
$65.00
$220.00
1
(1)
Fluphenazine Hydrochloride
Fluphenazine Hydrochloride is a dopamine D1 and D2 receptor antagonist that can bind to histamine H1
146-56-5 sc-205700
sc-205700A
sc-205700B
sc-205700C
1 g
5 g
50 g
100 g
$86.00
$224.00
$835.00
$1,215.00
0
(0)
Lidocaine
Lidocaine is a selective inverse peripheral histamine H1-receptor agonist
137-58-6 sc-204056
sc-204056A
50 mg
1 g
$49.00
$125.00
0
(0)
Cyproheptadine hydrochloride
Cyproheptadine hydrochloride is a non-selective 5-HT2 antagonist
969-33-5 sc-203557
50 mg
$85.00
2
(0)
Brompheniramine Maleate
Brompheniramine Maleate is a histamine H1 receptors antagonist
980-71-2 sc-210967
sc-210967A
25 mg
250 mg
$60.00
$200.00
1
(1)
Doxepin hydrochloride
Doxepin hydrochloride is a highly potent histamine H1 antagonist with affinity to H4 receptor
1229-29-4 sc-203930
1 g
$50.00
0
(1)
Hydroxyzine Dihydrochloride
Hydroxyzine Dihydrochloride is a hetercyclic H1 receptor antagonist
2192-20-3 sc-205716
sc-205716A
5 g
10 g
$75.00
$103.00
0
(0)
Antazoline hydrochloride
Antazoline hydrochloride is an anticholinergic and antihistamine agent
2508-72-7 sc-203515
sc-203515A
sc-203515B
100 mg
1 g
5 g
$65.00
$80.00
$200.00
0
(1)
Fenspiride Hydrochloride
Fenspiride Hydrochloride is an α adrenergic and H1 histamine receptor antaonist
5053-08-7 sc-207684
10 mg
$145.00
0
(0)
trans-Triprolidine hydrochloride
trans-Triprolidine hydrochloride is a potent H1 receptor antagonist
6138-79-0 sc-204354
1 g
$35.00
0
(1)
Clemastine fumarate
Clemastine fumarate is a selective histamine H1 antagonist
14976-57-9 sc-203897
100 mg
$95.00
0
(1)
Zotepine
Zotepine is an SR-2A and D2DR inhibitor and Histamine H1 receptor antagonist
26615-21-4 sc-360895
sc-360895A
10 mg
50 mg
$66.00
$246.00
3
(1)
Oxatomide
Oxatomide is an H1-histamine receptor antagonist
60607-34-3 sc-208136
10 mg
$200.00
0
(0)
Azelastine HCl
Azelastine HCl is an H1-receptor antagonist with antiallergic effects and disrupts TNF alpha activity
79307-93-0 sc-201096
sc-201096A
sc-201096B
sc-201096C
sc-201096D
100 mg
250 mg
1 g
5 g
10 g
$92.00
$200.00
$642.00
$1,950.00
$3,200.00
0
(1)
Levocabastine Hydrochloride
Levocabastine Hydrochloride is a histamine H1 receptor antagonist and anti-allergic agent
79547-78-7 sc-201095
10 mg
$184.00
4
(1)
Cetirizine Dihydrochloride
Cetirizine Dihydrochloride is a Histamine H1 receptor inverse agonist
83881-52-1 sc-202992
50 mg
$59.00
0
(0)
Mirtazapine
Mirtazapine is a potent SR-2, SR-3, and Histamine H1 receptor antagonist
85650-52-8 sc-204088
sc-204088A
10 mg
50 mg
$105.00
$409.00
0
(1)
Ebastine
Ebastine is an antagonist of the histamine H1-receptor
90729-43-4 sc-205663
sc-205663A
1 g
5 g
$104.00
$420.00
2
(1)
Pemirolast Potassium Salt
Pemirolast Potassium Salt is an inhibitor of mast cell mediator release
100299-08-9 sc-208156
10 mg
$165.00
0
(0)
Desloratadine
Desloratadine is a potent and selective H1-receptor agonist
100643-71-8 sc-202133
sc-202133A
100 mg
500 mg
$85.00
$384.00
3
(1)
Olopatadine Hydrochloride
Olopatadine Hydrochloride is a dual acting histamine H1-receptor antagonist and mast cell stabilizer
140462-76-6 sc-212473
25 mg
$140.00
0
(0)
(S)-Azelastine Hydrochloride
(S)-Azelastine Hydrochloride is n orally active Histamine H1 Receptor
153408-27-6 sc-208363
1 mg
$250.00
0
(0)
(R)-Azelastine Hydrochloride
An orally active Histamine H1 Receptor
153408-28-7 sc-208236
1 mg
$250.00
0
(0)
Fexofenadine HCl
Fexofenadine HCl is an antihistamine that inhibits Cox-1, Cox-2, and is a histamine H1 receptor agonist
153439-40-8 sc-203047
sc-203047A
10 mg
50 mg
$95.00
$399.00
0
(0)
Asenapine maleate
Asenapine maleate is An antagonist of noradrenalin, dopamine, 5-HT and receptors
65576-45-6 sc-361110
sc-361110A
10 mg
50 mg
$145.00
$615.00
0
(0)
Iso Loratadine
Iso Loratadine is an isomer of loratadine used to prepare tricyclic amides and ureas
170727-59-0 sc-394085
5 mg
$300.00
0
(0)
4-Diphenylmethoxy-1-methylpiperidine hydrochloride
4-Diphenylmethoxy-1-methylpiperidine hydrochloride is n inhibitor of Histamine H1 Receptor
132-18-3 sc-254657
10 g
$67.00
0
(0)
Mianserin hydrochloride
Mianserin hydrochloride is a non-selective 5-HT2 receptor antagonist with moderate affinity for 5-HT6
21535-47-7 sc-358986
100 mg
$105.00
1
(1)
Phenindamine Hydrochloride
Phenindamine Hydrochloride is a Histamine H1 receptor inhibitor
5503-08-2 sc-460196
50 mg
$280.00
0
(0)
Fexofenadine
Fexofenadine is A metabolite of of terfenadine, a H1-Histamine receptor antagonist
83799-24-0 sc-218475
100 mg
$200.00
1
(0)
Chlorpheniramine Maleate
Chlorpheniramine Maleate is an antagonist of the histamine H1-receptor
113-92-8 sc-204684
sc-204684A
5 g
25 g
$29.00
$49.00
1
(1)
(S)-Cetirizine Dihydrochloride
(S)-Cetirizine Dihydrochloride is a nonsedating type histamine H1-receptor antagonist
163837-48-7 sc-208364
2.5 mg
$250.00
0
(0)
Olopatadine N-Oxide
Olopatadine N-Oxide is an active metabolite of Olopatadine
203188-31-2 sc-212474
2.5 mg
$280.00
0
(0)
Fexofenadine-d6
Fexofenadine-d6 is a H1-Histamine receptor antagonist
548783-71-7 sc-211506
1 mg
$210.00
2
(0)
Doxylamine Succinate
Doxylamine Succinate is a H1 histamine receptor antagonist
562-10-7 sc-211381
100 mg
$100.00
1
(0)
Epinastine Hydrochloride
Epinastine Hydrochloride is a tetracyclic, histamine H1 receptor antagonist
108929-04-0 sc-211420
10 mg
$86.00
0
(0)
Azelastine-13C,d3
Azelastine-13C,d3 is A H1-histamine receptor antagonist
58581-89-8 (unlabeled) sc-217683
1 mg
$250.00
0
(0)
Rupatadine Fumarate
Rupatadine Fumarate is a dual histamine H1 and PAF antagonist
182349-12-8 sc-212795
10 mg
$160.00
0
(1)
Diphenhydramine-d6 Hydrochloride
Diphenhydramine-d6 Hydrochloride is a labeled H1-Histamine receptor antagonist
147-24-0 (unlabeled) sc-218244
1 mg
$250.00
0
(0)
Loratadine-d4
Loratadine-d4 is a labelled histamine H1-receptor inhibitor
381727-27-1 sc-280929
1 mg
$300.00
0
(1)
Chlorprothixene Hydrochloride
Chlorprothixene Hydrochloride is a D2DR inhibitor
6469-93-8 sc-211077
1 g
$30.00
1
(1)
Hydroxyzine
Hydroxyzine is an H1 receptor antagonist
68-88-2 sc-207748
500 mg
$240.00
0
(1)
Orphenadrine Citrate Salt
Orphenadrine Citrate Salt is a histaminergic compound
4682-36-4 sc-212481
5 g
$45.00
0
(0)
Promethazine Hydrochloride
Promethazine Hydrochloride is an antagonist of the histamine H1-receptor
58-33-3 sc-212586A
sc-212586
50 mg
100 mg
$70.00
$90.00
0
(1)
rac-N-Demethyl dimethindene-d3 hydrobromide
CAS: 151562-10-6 (unlabeled free base), MF: C19H19D3N2•HBr, MW: 362.32
151562-10-6 (unlabeled free base) sc-500664
1 mg
$280.00
0
(0)
Astemizole-d3
Astemizole-d3 is a labeled histamine H1-receptor anatagonist
1189961-39-4 sc-217667
1 mg
$450.00
0
(0)
Cetirizine-d8, Dihydrochloride
Cetirizine-d8, Dihydrochloride is A nonsedating type histamine H1-receptor antagonist
2070015-04-0 sc-217874
1 mg
$285.00
0
(0)
alpha-Hydroxy olopatadine
α-Hydroxy olopatadine is an inhibitor of Histamine H1 Receptor.
1331822-32-2 sc-489117
1 mg
$300.00
0
(0)
Hydroxyzine-d8 Dihydrochloride
Hydroxyzine-d8 Dihydrochloride is a H1 receptor antagonist
sc-280807
1 mg
$300.00
0
(0)
Hydroxyzine-d8
Hydroxyzine-d8 is a H1 receptor antagonist
68-88-2 (unlabeled) sc-280806
1 mg
$165.00
0
(0)
Olopatadine-d6 Hydrochloride
Olopatadine-d6 Hydrochloride is a labeled Olopatadine
1217229-05-4 sc-219484
1 mg
$280.00
0
(0)
Trimipramine-d3 Maleate Salt
Trimipramine-d3 Maleate Salt is a serotonin transport blocker that also blocks norepinephrine uptake
521-78-8 (unlabeled) sc-220342
1 mg
$200.00
0
(0)
Mebhydroline 1,5-naphthalenedisulfonate salt
Mebhydroline 1,5-naphthalenedisulfonate salt is a H1 histamine receptor antagonist
6153-33-9 sc-263459
1 g
$20.00
0
(0)
Desmethyl Nizatidine
Desmethyl Nizatidine is a main metabolite of Nizatidine
82586-78-5 sc-391545
2.5 mg
$280.00
0
(0)
Acrivastine
Acrivastine is a second-generation antihistamine
87848-99-5 sc-357283
sc-357283A
10 mg
50 mg
$100.00
$304.00
0
(0)
Pheniramine maleate salt
Pheniramine maleate salt is A H1 histamine receptor antagonist
132-20-7 sc-253258
5 g
$110.00
0
(0)
Bepotastine besilate
Bepotastine besilate is an inhibitor of Histamine H1 Receptor.
190786-44-8 sc-482068
10 mg
$79.00
0
(0)
Desmethyl doxylamine
1221-70-1 sc-500284
sc-500284A
100 mg
1 g
$300.00
$2,400.00
0
(0)
Diphenylamine Hydrochloride
Diphenylamine Hydrochloride is a antagonist of histamine H1 receptor
537-67-7 sc-485023
25 g
$68.00
0
(0)