p300 Activators
Items 1 to 10 of 11 total
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| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
CTPB | 586976-24-1 | sc-202558 sc-202558A | 1 mg 5 mg | $59.00 $165.00 | 4 | |
CTPB functions as a selective p300 inhibitor, exhibiting unique interactions with the acetyltransferase domain. Its structural conformation allows for precise binding, disrupting the enzyme's catalytic activity. This inhibition alters histone acetylation patterns, influencing gene expression regulation. The compound's kinetic profile reveals a rapid association and dissociation with p300, underscoring its potential to modulate transcriptional dynamics in cellular environments. | ||||||
C646 | 328968-36-1 | sc-364452 sc-364452A | 10 mg 50 mg | $265.00 $944.00 | 5 | |
C646 is a competitive inhibitor of p300 that binds to its acetyl-CoA binding site. Although primarily known as an inhibitor, it might indirectly activate p300 by preventing it from binding to molecules that inhibit its function. | ||||||
Anacardic Acid | 16611-84-0 | sc-202463 sc-202463A | 5 mg 25 mg | $102.00 $204.00 | 13 | |
Anacardic Acid is found in the shell of the cashew nut. It has been shown to stimulate p300, which in turn enhances histone acetylation. Histone acetylation is a process that opens up the chromatin structure, enhancing gene transcription. | ||||||
Curcumin | 458-37-7 | sc-200509 sc-200509A sc-200509B sc-200509C sc-200509D sc-200509F sc-200509E | 1 g 5 g 25 g 100 g 250 g 1 kg 2.5 kg | $37.00 $69.00 $109.00 $218.00 $239.00 $879.00 $1968.00 | 47 | |
Curcumin is the active component of turmeric. It has been demonstrated to increase the activity of p300/CBP, which can lead to increased histone acetylation and gene transcription. | ||||||
Brassinolide | 72962-43-7 | sc-391736 sc-391736A | 2 mg 10 mg | $106.00 $339.00 | 2 | |
Brassinolide is a plant steroid that has been shown to enhance the expression and function of p300, thereby enhancing histone acetylation and gene transcription. | ||||||
Resveratrol | 501-36-0 | sc-200808 sc-200808A sc-200808B | 100 mg 500 mg 5 g | $80.00 $220.00 $460.00 | 64 | |
Resveratrol is a polyphenolic compound found in various fruits such as grapes and some berries. It has been shown to increase the acetyltransferase activity of p300, which can lead to increased histone acetylation and gene transcription. | ||||||
(−)Epicatechin | 490-46-0 | sc-205672 sc-205672A | 1 mg 5 mg | $51.00 $138.00 | ||
This is a flavonoid, common in cocoa, tea, and some fruits. It has been suggested to enhance p300 activity, though the exact mechanism is not fully understood. It may increase acetylation and subsequent gene transcription. | ||||||
D,L-Sulforaphane | 4478-93-7 | sc-207495A sc-207495B sc-207495C sc-207495 sc-207495E sc-207495D | 5 mg 10 mg 25 mg 1 g 10 g 250 mg | $153.00 $292.00 $489.00 $1325.00 $8465.00 $933.00 | 22 | |
This compound is found in cruciferous vegetables such as broccoli. It has been demonstrated to increase the activity of p300, which can lead to increased histone acetylation and gene transcription. | ||||||
Lycopene | 502-65-8 | sc-205738 sc-205738A sc-205738B | 1 mg 5 mg 1 g | $146.00 $582.00 $6248.00 | 4 | |
Lycopene is a carotenoid found in tomatoes. It has been suggested to enhance the activity of p300, possibly increasing histone acetylation and gene transcription. | ||||||
Quercetin | 117-39-5 | sc-206089 sc-206089A sc-206089E sc-206089C sc-206089D sc-206089B | 100 mg 500 mg 100 g 250 g 1 kg 25 g | $11.00 $17.00 $110.00 $250.00 $936.00 $50.00 | 33 | |
This flavonoid, found in many fruits and vegetables, has been suggested to enhance p300 activity, potentially increasing histone acetylation and gene transcription. | ||||||