GPR54 Activators
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Items 1 to 10 of 11 total
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| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
Metastin | sc-221884 | 500 µg | $310.00 | |||
Metastin is a selective GPR54 activator known for its unique ability to stabilize receptor conformation through specific ligand-receptor interactions. This compound promotes receptor oligomerization, which is crucial for initiating intracellular signaling cascades. Its distinct structural motifs enhance binding affinity, leading to accelerated activation kinetics. Additionally, Metastin's hydrophilic characteristics facilitate effective membrane permeability, influencing its bioavailability and interaction with GPR54. | ||||||
Metastin (45-54) | 374675-21-5 | sc-221883 sc-221883A sc-221883B | 1 mg 20 mg 60 mg | $112.00 $1457.00 $6000.00 | 2 | |
Metastin (45-54) is a potent GPR54 activator characterized by its ability to induce conformational changes in the receptor, enhancing downstream signaling pathways. Its unique peptide sequence allows for high specificity in binding, promoting receptor dimerization and subsequent activation. The compound exhibits rapid kinetics, facilitating swift cellular responses. Furthermore, its structural features contribute to favorable interactions with lipid membranes, optimizing its functional efficacy in cellular environments. | ||||||
Clomiphene Citrate | 50-41-9 | sc-205636 sc-205636A | 1 g 5 g | $84.00 $176.00 | 1 | |
By modulating luteinizing hormone and follicle-stimulating hormone levels, this compound may have an impact on GPR54 signaling. | ||||||
Tamoxifen | 10540-29-1 | sc-208414 | 2.5 g | $272.00 | 18 | |
It may influence the expression or signaling of GPR54 by modulating estrogenic activity. | ||||||
Medroxyprogesterone 17-Acetate | 71-58-9 | sc-205744 sc-205744A | 500 mg 1 g | $67.00 $99.00 | ||
Could potentially influence GPR54 activity by interacting with progesterone receptors and modulating related signaling pathways. | ||||||
MDV3100 | 915087-33-1 | sc-364354 sc-364354A | 5 mg 50 mg | $245.00 $1051.00 | 7 | |
By modulating androgenic activity, it may affect the signaling or expression of GPR54. | ||||||
Forskolin | 66575-29-9 | sc-3562 sc-3562A sc-3562B sc-3562C sc-3562D | 5 mg 50 mg 1 g 2 g 5 g | $78.00 $153.00 $740.00 $1413.00 $2091.00 | 73 | |
By increasing cAMP levels, it might influence the signaling cascades associated with GPR54. | ||||||
Dibutyryl-cAMP | 16980-89-5 | sc-201567 sc-201567A sc-201567B sc-201567C | 20 mg 100 mg 500 mg 10 g | $47.00 $136.00 $492.00 $4552.00 | 74 | |
Activating protein kinase A might modulate the phosphorylation states of proteins in GPR54-related pathways. | ||||||
Verapamil | 52-53-9 | sc-507373 | 1 g | $374.00 | ||
By modifying intracellular calcium levels, it may influence GPR54 signaling. | ||||||
PMA | 16561-29-8 | sc-3576 sc-3576A sc-3576B sc-3576C sc-3576D | 1 mg 5 mg 10 mg 25 mg 100 mg | $41.00 $132.00 $214.00 $500.00 $948.00 | 119 | |
Modulating the activity of Protein Kinase C might influence the signaling pathways associated with GPR54. | ||||||