OCTN1 Inhibitors
Items 1 to 10 of 12 total
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| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
Quinidine | 56-54-2 | sc-212614 | 10 g | $102.00 | 3 | |
Quinidine, a stereoisomer of quinine, is known to inhibit OCTN1. It acts by competing for the transport sites, reducing the uptake of other substrates. | ||||||
Verapamil | 52-53-9 | sc-507373 | 1 g | $367.00 | ||
Verapamil, a calcium channel blocker, has been shown to inhibit OCTN1-mediated transport, likely by competing for binding sites. | ||||||
Mepyramine maleate | 59-33-6 | sc-203629 sc-203629A | 100 mg 1 g | $65.00 $220.00 | 1 | |
Pyrilamine, an antihistamine, can inhibit OCTN1. It likely interferes with the transporters ability to bind and translocate its natural substrates. | ||||||
Corticosterone | 50-22-6 | sc-300391 sc-300391A | 100 mg 500 mg | $57.00 $108.00 | 2 | |
Corticosterone is known to inhibit OCTN1. It may compete with other substrates for binding, thus reducing the transport efficiency of OCTN1. | ||||||
Metformin-d6, Hydrochloride | 1185166-01-1 | sc-218701 sc-218701A sc-218701B | 1 mg 5 mg 10 mg | $286.00 $806.00 $1510.00 | 1 | |
Metformin has been found to inhibit OCTN1, potentially by competitive inhibition at the substrate binding site. | ||||||
Cimetidine | 51481-61-9 | sc-202996 sc-202996A | 5 g 10 g | $62.00 $86.00 | 1 | |
Cimetidine, a histamine H2 receptor antagonist, can inhibit OCTN1 by competing for the cationic transport pathway. | ||||||
Propranolol | 525-66-6 | sc-507425 | 100 mg | $180.00 | ||
Propranolol, a beta-blocker, is capable of inhibiting OCTN1. Its interaction with OCTN1 can affect the disposition of other drugs. | ||||||
Levofloxacin | 100986-85-4 | sc-252953 sc-252953B sc-252953A | 10 mg 250 mg 1 g | $39.00 $45.00 $53.00 | 3 | |
Levofloxacin, a fluoroquinolone antibiotic, has been reported to inhibit OCTN1, potentially affecting the pharmacokinetics of co-administered drugs. | ||||||
Procainamide hydrochloride | 614-39-1 | sc-202297 | 10 g | $52.00 | ||
Procainamide, an antiarrhythmic agent, inhibits OCTN1. It competes with other substrates, influencing the transport of organic cations. | ||||||
Disopyramide | 3737-09-5 | sc-207585 | 100 mg | $340.00 | ||
Disopyramide, another antiarrhythmic drug, has been shown to inhibit OCTN1, affecting the transporter′s function. | ||||||