CB1 Activators
Items 1 to 10 of 25 total
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| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
Rimonabant | 168273-06-1 | sc-205491 sc-205491A | 5 mg 10 mg | $72.00 $160.00 | 15 | |
Rimonabant is a selective antagonist of the CB1 receptor, characterized by its unique ability to disrupt endocannabinoid signaling. Its molecular structure allows for specific interactions with the receptor's binding pocket, leading to conformational changes that inhibit downstream signaling pathways. This compound exhibits distinct kinetic profiles, influencing receptor desensitization and internalization, thereby modulating neurotransmitter release and synaptic plasticity in neural circuits. | ||||||
Magnolol | 528-43-8 | sc-204797 sc-204797A | 5 mg 25 mg | $42.00 $185.00 | 1 | |
Magnolol acts as a modulator of the CB1 receptor, showcasing a unique affinity for specific allosteric sites that influence receptor dynamics. Its molecular interactions promote subtle conformational shifts, enhancing or diminishing receptor activity. This compound exhibits intriguing reaction kinetics, affecting the rate of receptor activation and desensitization. Additionally, its hydrophobic characteristics facilitate membrane penetration, impacting cellular signaling pathways and lipid interactions. | ||||||
Oleamide | 301-02-0 | sc-358696 sc-358696A sc-358696B sc-358696C sc-358696D | 10 mg 25 mg 50 mg 100 mg 500 mg | $60.00 $71.00 $122.00 $214.00 $627.00 | ||
Oleamide is a fascinating compound that interacts with the CB1 receptor, exhibiting a unique ability to stabilize receptor conformations through hydrogen bonding and hydrophobic interactions. Its presence can modulate the receptor's signaling efficiency, influencing downstream pathways. The compound's lipid-like properties enhance its integration into cellular membranes, potentially altering membrane fluidity and affecting receptor localization. This interplay can lead to distinct physiological responses, showcasing its role in cellular communication. | ||||||
Leelamine HCl | 1446-61-3 | sc-200375 sc-200375A | 10 mg 50 mg | $124.00 $530.00 | ||
Leelamine HCl is a notable compound that engages with the CB1 receptor, characterized by its ability to form ionic and dipole-dipole interactions, which can significantly influence receptor activation. Its unique structural features allow it to traverse lipid bilayers efficiently, impacting membrane dynamics and receptor accessibility. Additionally, Leelamine HCl may alter the kinetics of receptor-ligand binding, potentially leading to varied signaling outcomes and cellular responses. | ||||||
ABN-CBD | 22972-55-0 | sc-203488A sc-203488B sc-203488 sc-203488C | 1 mg 5 mg 10 mg 25 mg | $36.00 $143.00 $235.00 $541.00 | 1 | |
ABN-CBD is a distinctive compound that interacts with the CB1 receptor through a combination of hydrophobic and hydrogen bonding interactions, enhancing its binding affinity. Its unique conformation facilitates selective receptor engagement, potentially influencing downstream signaling pathways. The compound's ability to modulate receptor conformational states may lead to altered signal transduction dynamics, affecting cellular behavior and response patterns in complex biological systems. | ||||||
Olvanil | 58493-49-5 | sc-201454 sc-201454A | 5 mg 25 mg | $47.00 $201.00 | 1 | |
Olvanil exhibits a unique binding profile with the CB1 receptor, characterized by its ability to form specific hydrophobic pockets and engage in van der Waals interactions. This compound's structural flexibility allows it to adopt conformations that stabilize receptor activation, influencing allosteric modulation. Its kinetic properties suggest a rapid association and dissociation with the receptor, potentially leading to nuanced effects on intracellular signaling cascades and receptor desensitization mechanisms. | ||||||
CP-55,940 | 83002-04-4 | sc-200359 sc-200359A | 5 mg 25 mg | $185.00 $850.00 | 4 | |
CP-55,940 demonstrates a remarkable affinity for the CB1 receptor, engaging in intricate hydrogen bonding and hydrophobic interactions that enhance its binding efficacy. Its unique stereochemistry facilitates selective receptor activation, promoting distinct signaling pathways. The compound's dynamic conformational changes contribute to its prolonged receptor engagement, influencing downstream effects on neurotransmitter release and cellular response mechanisms. This intricate interplay underscores its complex pharmacodynamics. | ||||||
Arvanil | 128007-31-8 | sc-202065 | 5 mg | $150.00 | 1 | |
Arvanil exhibits a unique binding profile with the CB1 receptor, characterized by its ability to form specific van der Waals interactions and electrostatic contacts. This compound's structural flexibility allows it to adopt multiple conformations, optimizing its fit within the receptor's binding pocket. The kinetic properties of Arvanil facilitate rapid receptor activation, leading to nuanced modulation of intracellular signaling cascades. Its distinct molecular interactions contribute to a complex landscape of receptor dynamics and functional outcomes. | ||||||
DEA | 150314-35-5 | sc-203024 | 5 mg | $56.00 | ||
DEA interacts with the CB1 receptor through a combination of hydrophobic and hydrogen bonding interactions, enhancing its affinity and selectivity. Its unique steric configuration allows for effective spatial orientation within the receptor, promoting efficient signal transduction. The compound's reactivity as an acid halide enables it to participate in nucleophilic attack mechanisms, influencing downstream pathways. This dynamic interplay of molecular forces shapes its role in receptor-mediated processes. | ||||||
(R)-Methanandamide | 157182-49-5 | sc-200792 sc-200792A | 5 mg 25 mg | $56.00 $175.00 | 1 | |
(R)-Methanandamide exhibits a distinctive binding profile with the CB1 receptor, characterized by its ability to form multiple van der Waals interactions that stabilize the receptor-ligand complex. Its chiral nature contributes to a specific orientation that enhances receptor activation. Additionally, the compound's structural flexibility allows it to adapt to conformational changes in the receptor, facilitating a robust signaling cascade. This interplay of molecular dynamics is crucial for its functional efficacy. | ||||||