PI 3-kinase Inhibitors

Santa Cruz Biotechnology now offers a broad range of PI 3-kinase Inhibitors. Phosphatidylinositol 3-kinase (PI 3-kinase) phosphorylates the 3' OH position of the inositol ring of inositol lipids and is composed of p85 and p110 subunits. PI 3-kinase Inhibitors offered by Santa Cruz inhibit PI 3-kinase and, in some cases, other cell survival and glucose regulation related proteins. View detailed PI 3-kinase Inhibitor specifications, including PI 3-kinase Inhibitor CAS number, molecular weight, molecular formula and chemical structure, by clicking on the product name.

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PRODUCT NAME/Application CAS Catalog # QUANTITY Price Citations RATING
Wortmannin
Wortmannin is an antibiotic and fungal metabolite, able to selectively inhibit phosphatidylinositol 3-kinase.
19545-26-7 sc-3505
sc-3505A
sc-3505B
1 mg
5 mg
20 mg
$55.00
$205.00
$399.00
92
(3)
Piceatannol
Piceatannol is an inhibitor of Syk and NF-κB activation
10083-24-6 sc-200610
sc-200610A
sc-200610B
1 mg
5 mg
25 mg
$40.00
$62.00
$186.00
11
(2)
Thioridazine Hydrochloride
Thioridazine Hydrochloride is a D2DR, D4DR, and calcium channel protein inhibitor
130-61-0 sc-201149A
sc-201149
sc-201149C
sc-201149D
sc-201149B
5 mg
1 g
25 g
100 g
5 g
$20.00
$47.00
$400.00
$1,200.00
$100.00
0
(1)
LY 294002
LY 294002 is a potent blocker of PI 3-kinase/Akt signaling
154447-36-6 sc-201426
sc-201426A
5 mg
25 mg
$119.00
$384.00
136
(1)
LY 303511
LY 303511 is a negative control for PI 3-kinase inhibitors
154447-38-8 sc-202215
sc-202215A
1 mg
5 mg
$65.00
$268.00
3
(1)
Hypericin
Hypericin is a Protein Kinase C, CKII, MAP, Insulin R, EGFR, and PI-3 kinase inhibitor with antiviral activity.
548-04-9 sc-3530
sc-3530A
1 mg
5 mg
$58.00
$200.00
10
(1)
IC-87114
IC-87114 is a PI3K inhibitor with action against fMLP-PIP3
371242-69-2 sc-364509
sc-364509A
5 mg
50 mg
$140.00
$1,060.00
1
(1)
Myricetin
Myricetin is a cell-permeable, ATP-competitive inhibitor of various casein kinases and protein kinases.
529-44-2 sc-203147
sc-203147A
sc-203147B
sc-203147C
sc-203147D
25 mg
100 mg
1 g
25 g
100 g
$93.00
$180.00
$250.00
$490.00
$982.00
2
(1)
PIK-75, free base
PIK-75, free base is a free base is a selective inhibitor of PI 3-kinase p110α
372196-67-3 sc-394297
5 mg
$81.00
1
(0)
XL-147 derivative 2
XL-147 derivative 2 is an ATP-competetive class I PI3K inhibitor
956958-53-5 sc-364658
sc-364658A
10 mg
50 mg
$255.00
$700.00
1
(0)
Toyocamycin
Toyocamycin is an antimetabolite with a broad spectrum of antibiotic activity
606-58-6 sc-362812
10 mg
$98.00
0
(1)
WHI-P 154
WHI-P 154 is a JAK3 inhibitor which inhibits other common kinases
211555-04-3 sc-204395
sc-204395A
10 mg
50 mg
$109.00
$615.00
3
(1)
CAL-101
CAL-101 is a potent PI3K p110δ inhibitor
870281-82-6 sc-364453
10 mg
$180.00
2
(1)
GSK2126458
GSK2126458 is an inhibitor of p110 mutants
1086062-66-9 sc-364503
sc-364503A
2 mg
10 mg
$255.00
$1,009.00
0
(0)
Fisetin
Fisetin is a potent sirtuin activating compound (STAC), antiinflammatory and anticancer agent
528-48-3 sc-276440
sc-276440A
sc-276440B
sc-276440C
sc-276440D
50 mg
100 mg
500 mg
1 g
100 g
$50.00
$75.00
$100.00
$150.00
$2,800.00
6
(1)
17beta-hydroxy Wortmannin
17β-hydroxy Wortmannin is an inhibitor of recombinant PI 3-kinase and mTOR
58053-83-1 sc-358740
sc-358740A
500 µg
1 mg
$92.00
$176.00
0
(1)
Miltefosine
Miltefosine is a PI 3-kinase and Akt inhibitor that also inhibits anti-IgE induced histamine release
58066-85-6 sc-203135
50 mg
$73.00
7
(1)
SF1126
SF1126 is a prodrug containing the pan-PI3K/mTOR inhibitor LY294002/SF1101
936487-67-1 sc-391584
sc-391584A
5 mg
10 mg
$700.00
$1,300.00
7
(0)
CH5132799
CH5132799 is a PI3K and FRAP inhibitor
1007207-67-1 sc-364460
sc-364460A
5 mg
50 mg
$360.00
$1,650.00
0
(0)
AS-252424
AS-252424 is a selective PI 3-kinase p110γ inhibitor
900515-16-4 sc-202961
sc-202961A
1 mg
5 mg
$40.00
$152.00
0
(1)
LY 294002, 4′-NH2
LY 294002, 4′-NH2 is a PI 3-kinase inhibitor
942289-87-4 sc-203121
sc-203121A
5 mg
50 mg
$153.00
$772.00
1
(1)
(±)-Naringenin
(±)-Naringenin is a PI 3-kinase inhibitor
67604-48-2 sc-203155
sc-203155A
sc-203155B
sc-203155C
sc-203155D
1 g
5 g
25 g
100 g
500 g
$40.00
$80.00
$150.00
$300.00
$800.00
1
(1)
PI 3-Kbeta Inhibitor VI, TGX-221
PI 3-Kβ Inhibitor VI, TGX-221 is a reversible ATP-competitive inhibitor of PI 3-kinase β
663619-89-4 sc-203190
1 mg
$437.00
0
(0)
PI 3-Kgamma Inhibitor
PI 3-Kγ Inhibitor is a cell-permeable, potent, selective, and ATP-competitive inhibitor of PI 3-kinase
648450-29-7 sc-203191
5 mg
$76.00
0
(0)
CAY10505
CAY10505 is a PI3K inhibitor
1218777-13-9 sc-364456
sc-364456A
10 mg
50 mg
$80.00
$280.00
0
(0)
PI-103
PI-103 is an ATP-competitive DNA-PK, PI 3-kinase, and FRAP inhibitor
371935-74-9 sc-203193
sc-203193A
1 mg
5 mg
$31.00
$125.00
3
(1)
YM201636
YM201636 is a selective, potent inhibitor of phosphatidylinositol phosphate kinase PIKfyve that can completely block PI 3-kinase activation.
371942-69-7 sc-204193
5 mg
$199.00
5
(1)
Autophagy Inhibitor, 3-MA
Autophagy Inhibitor, 3-MA is a multi-use inhibitor that inhibits autophagy by blocking autophagosome formation via the inhibition of type III Phosphatidylinositol 3-kinases.
5142-23-4 sc-205596
sc-205596A
50 mg
500 mg
$50.00
$250.00
105
(3)
LY-294,002 hydrochloride
LY-294,002 hydrochloride is a highly selective inhibitor of PI 3-kinase
934389-88-5 sc-215273
sc-215273A
1 mg
5 mg
$65.00
$151.00
3
(1)
Quercetin
Quercetin is a PI 3-kinase inhibitor, GPR30 activator, and apoptosis inducer
117-39-5 sc-206089
sc-206089A
sc-206089B
sc-206089E
sc-206089C
sc-206089D
100 mg
500 mg
25 g
100 g
250 g
1 kg
$10.00
$15.00
$39.00
$100.00
$240.00
$900.00
24
(2)
3prime,4prime,7-Trihydroxyisoflavone
3′,4′,7-Trihydroxyisoflavone is an inhibitor of β-galactosidase enzyme
485-63-2 sc-206722
200 mg
$255.00
0
(1)
Compound 15e
Compound 15e is a potent inhibitor of the PI 3-kinase p110α isoform
371943-05-4 sc-202551
sc-202551A
1 mg
5 mg
$51.00
$206.00
0
(0)
PIK-90
PIK-90 is a selective inhibitor of PI3K isoforms
677338-12-4 sc-364587
sc-364587A
5 mg
50 mg
$105.00
$555.00
0
(0)
PIK-294
PIK-294 is a selective PI3K inhibitor
900185-02-6 sc-364586
sc-364586A
5 mg
50 mg
$309.00
$1,764.00
0
(0)
GSK 1059615
GSK 1059615 is a potent inhibitor of PI 3-kinase and FRAP (mTOR)
958852-01-2 sc-361198
sc-361198A
10 mg
50 mg
$179.00
$825.00
0
(0)
PP121
PP121 is an inhibitor of c-Abl, PI 3-kinase, PDGFR, Hck, FRAP, Flk-1, SRC, and DNA-PK
1092788-83-4 sc-301605
5 mg
$139.00
1
(0)
PI 3-Kalpha Inhibitor VIII
PI 3-Kα Inhibitor VIII is a potent PI 3-kinase inhibitor
372196-77-5 sc-364583
5 mg
$440.00
0
(0)
PIK-293
PIK-293 is a PI3K inhibitor
900185-01-5 sc-364585
sc-364585A
5 mg
50 mg
$370.00
$1,950.00
0
(0)
BYL719
BYL719 is a selective inhibitor of phosphoinositide 3-kinase α (PI3Kα), equipotent against wild type and mutant isoforms.
1217486-61-7 sc-391001
sc-391001A
sc-391001B
sc-391001C
sc-391001D
sc-391001E
5 mg
10 mg
50 mg
100 mg
500 mg
1 g
$370.00
$568.00
$720.00
$1,140.00
$4,800.00
$9,000.00
1
(0)
PI3K/HDAC Inhibitor
PI3K/HDAC Inhibitor is an inhibitor of HDAC1, HDAC2, HDAC3, HDAC6, HDAC8, HDAC10, and HDAC11
1339928-25-4 sc-364584
sc-364584A
5 mg
10 mg
$340.00
$462.00
0
(0)
N-Acetyl-Asp-Tyr(2-malonyl)-Val-Pro-Met-Leu-NH2
N-Acetyl-Asp-Tyr(2-malonyl)-Val-Pro-Met-Leu-NH2 is a protein tyrosine kinase inhibitor
sc-364544
sc-364544A
1 mg
5 mg
$85.00
$415.00
0
(0)
N-Acetyl-Asp-Tyr(PO3H2)-Val-Pro-Met-Leu-NH2
N-Acetyl-Asp-Tyr(PO3H2)-Val-Pro-Met-Leu-NH2 is an effective protein tyrosine kinase inhibitor
sc-364545
1 mg
$62.00
0
(0)
Viridiol
Viridiol is a steroid antibiotic shown to be a PI 3-kinase inhibitor
23820-80-6 sc-391040A
sc-391040
250 µg
1 mg
$73.00
$180.00
0
(0)
Demethoxyviridiol
Demethoxyviridiol is A fungal metabolite and inhibitor of phosphatidylinositol 3-kinase
56617-66-4 sc-391780
1 mg
$250.00
0
(0)
AS-604850
AS-604850 is an ATP-competitive inhibitor of PI 3-kinase γ
648449-76-7 sc-221271
sc-221271A
1 mg
5 mg
$36.00
$130.00
0
(0)
AS-605240
AS-605240 is an inhibitor of PI 3-kinase γ
648450-29-7 sc-221272
sc-221272A
1 mg
5 mg
$23.00
$80.00
1
(1)
PI 3-Kalpha Inhibitor IV
PI 3-Kα Inhibitor IV is a potent and isoform-selective inhibitor of the PI 3-kinase family
sc-222170
5 mg
$215.00
1
(0)
AS 041164
AS 041164 is a potent inhibitor of PI 3-kinase
1146702-72-8 sc-291912
sc-291912A
1 mg
5 mg
$23.00
$65.00
0
(0)
BAG 956
BAG 956 is a dual PDK1 and class I PI 3-kinase inhibitor
853910-02-8 sc-291923
sc-291923A
10 mg
50 mg
$215.00
$906.00
0
(0)
TG 100713
TG 100713 is an inhibitor of PI3-kinase
925705-73-3 sc-362809
sc-362809A
10 mg
50 mg
$199.00
$849.00
0
(0)
NVP-BGT226
NVP-BGT226 is a novel dual PI 3-kinase/mTOR (FRAP) inhibitor
1245537-68-1 sc-364553
sc-364553A
5 mg
50 mg
$474.00
$1,874.00
0
(0)
PIK-75, hydrochloride
PIK-75, hydrochloride is a selective inhibitor of PI 3-kinase isoform p110α
372196-77-5 sc-296089
sc-296089A
1 mg
5 mg
$27.00
$120.00
0
(1)
PP242
PP242 is a selective FRAP inhibitor
1092351-67-1 sc-301606A
sc-301606
1 mg
5 mg
$55.00
$166.00
6
(1)
A66
A66 is an inhibitor for oncogenic forms of p110
1166227-08-2 sc-364394
sc-364394A
5 mg
50 mg
$255.00
$1,455.00
0
(0)
BEZ235
BEZ235 is a dual PI3K and mTOR inhibitor
915019-65-7 sc-364429
50 mg
$198.00
8
(1)
3-Methyl-d3-adenine
3-Methyl-d3-adenine is an isotope labeled DNA methylater
5142-23-4 (unlabeled) sc-216512
1 mg
$200.00
0
(0)
BIP-135
BIP-135 is a GSK-3 inibitor with modest efficacy against PKC and PI3K
941575-71-9 sc-364435
sc-364435A
5 mg
25 mg
$105.00
$410.00
0
(0)
BKM120
BKM120 is BKM120 is a PI 3-kinase family inhibitor
944396-07-0 sc-364437
sc-364437A
sc-364437B
sc-364437C
5 mg
10 mg
25 mg
50 mg
$170.00
$225.00
$270.00
$325.00
8
(0)
PX-866
PX-866 is a PI3K inhibitor
502632-66-8 sc-396764
sc-396764A
1 mg
5 mg
$89.00
$270.00
0
(1)
GDC-0941
GDC-0941 is a potent inhibitor the PI 3-kinase family
957054-30-7 sc-364498
sc-364498A
5 mg
10 mg
$180.00
$191.00
2
(1)
GDC-0980
GDC-0980 is a PI3K and FRAP (mTOR) kinase inhibitor
1032754-93-0 sc-364499
sc-364499A
5 mg
50 mg
$340.00
$1,400.00
0
(0)
PIK-93
PIK-93 is a novel and potent inhibitor
593960-11-3 sc-364588
5 mg
$255.00
0
(0)
TG100-115
TG100-115 is a PI3K and FRAP inhibitor with some action against Akt
677297-51-7 sc-364634
sc-364634A
5 mg
100 mg
$240.00
$1,800.00
1
(0)
Akt Inhibitor
Akt Inhibitor is a phosphatidylinositol ether analog that potently and selectively inhibits Akt
sc-394003
1 mg
$240.00
5
(1)
XL-147 derivative 1
XL-147 derivative 1 is a potent class I PI3K inhibitor
1349796-36-6 sc-364660
sc-364660A
5 mg
50 mg
$189.00
$1,725.00
0
(0)