GABA Receptor Inhibitors

Santa Cruz Biotechnology now offers a broad range of GABA Receptor Inhibitors. In the central nervous system GABA functions as the main inhibitory transmitter by increasing a Cl- conductance that inhibits neuronal firing. GABA has been shown to activate both ionotropic (GABAA) and metabotropic (GABAB) receptors as well as a third class of receptors called GABAC. GABA Receptor Inhibitors offered by Santa Cruz inhibit GABA Receptor and, in some cases, other ionotropic and metabotropic receptor related proteins. View detailed GABA Receptor Inhibitor specifications, including GABA Receptor Inhibitor CAS number, molecular weight, molecular formula and chemical structure, by clicking on the product name.

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PRODUCT NAME/Application CAS Catalog # QUANTITY Price Citations RATING
(-)-Bicuculline methobromide
(−)-Bicuculline methobromide is an N-methylated derivative of the GABAA antagonist bicuculline
73604-30-5 sc-200436
50 mg
$143.00
0
(1)
(-)-alpha-Thujone
(−)-α-Thujone is a GABAA antagonist and chiral building block
546-80-5 sc-252342
1 ml
$73.00
0
(0)
Pregnenolone
Pregnenolone is an prohormone neurosteroid also a precursor to gonadal steroid hormones and the adrenal corticosteroids
145-13-1 sc-204860
sc-204860A
sc-204860B
sc-204860C
5 g
25 g
100 g
500 g
$47.00
$83.00
$120.00
$425.00
0
(1)
NNC 711
NNC 711 is a potent and selective inhibitor of GABA T-1
145645-62-1 sc-204132
sc-204132A
5 mg
25 mg
$116.00
$301.00
0
(0)
CGP 54626 hydrochloride
CGP 54626 hydrochloride is a potent and selective GABA b receptor antagonist
149184-21-4 sc-361142
sc-361142A
10 mg
50 mg
$195.00
$0.00
0
(1)
Flumazenil (Ro 15-1788)
Flumazenil (Ro 15-1788) is a benzodiazepine antagonist
78755-81-4 sc-200161
sc-200161A
20 mg
100 mg
$62.00
$259.00
10
(1)
Picrotoxin
Picrotoxin is a GABAA receptor antagonist
124-87-8 sc-202765
sc-202765A
sc-202765B
1 g
5 g
25 g
$60.00
$270.00
$1,270.00
4
(2)
CGP 35348
CGP 35348 is a selective GABAB receptor antagonist
123690-79-9 sc-361138
sc-361138A
10 mg
50 mg
$169.00
$681.00
0
(1)
SR 95531 Hydrobromide
SR 95531 Hydrobromide is a selective GABAA receptor antagonist
104104-50-9 sc-203701
sc-203701A
10 mg
50 mg
$145.00
$490.00
0
(1)
(+)-Bicuculline
(+)-Bicuculline is a GABA A receptor antagonist
485-49-4 sc-202498
sc-202498A
50 mg
250 mg
$54.00
$201.00
0
(1)
CGP 52432
CGP 52432 is A selective and effective GABAB receptor antagonist
139667-74-6 sc-361141
sc-361141A
10 mg
50 mg
$199.00
$825.00
0
(0)
Furosemide
Furosemide is an inhibitor of NKCC and a GABAA receptor antagonist
54-31-9 sc-203961
50 mg
$39.00
0
(1)
(-)-Bicuculline methiodide
(−)-Bicuculline methiodide is a N-methylated derivative of the GABAA antagonist (+)-bicuculline
40709-69-1 sc-200485
50 mg
$142.00
5
(1)
TPMPA
TPMPA is TPMPA is a competitive, selective GABAC antagonist
182485-36-5 sc-204352
sc-204352A
10 mg
50 mg
$215.00
$750.00
1
(0)
Propybicyphat
Propybicyphat is a GABA-gated chloride channel blocker
51486-74-9 sc-301615
1 mg
$229.00
0
(0)
(+)-Tubocurarine dichloride
(+)-Tubocurarine Hydrochloride is a neuromuscular block inducer
57-94-3 sc-202845
50 mg
$69.00
0
(0)
Thiocolchicoside
Thiocolchicoside is a GABAA receptor antagonist
602-41-5 sc-202839
sc-202839A
1 mg
5 mg
$30.00
$120.00
0
(0)
Pregnenolone sulfate sodium salt
Pregnenolone sulfate sodium salt is is a GABAA receptor antagonist
1852-38-6 sc-301609
50 mg
$60.00
1
(1)
Cyclothiazide
Cyclothiazide is a potent inhibitor of desensitization of AMPA receptors
2259-96-3 sc-202560
sc-202560A
10 mg
50 mg
$75.00
$208.00
0
(1)
Guvacine hydrochloride
Guvacine hydrochloride is inhibits GABA uptake
6027-91-4 sc-263347
25 mg
$93.00
0
(1)
Riluzole
Riluzole is a sodium channel protein inhibitor
1744-22-5 sc-201081
sc-201081A
sc-201081B
sc-201081C
20 mg
100 mg
1 g
25 g
$15.00
$180.00
$200.00
$300.00
0
(1)
Bilobalide
Bilobalide is a compound with neuroprotective, antibacterial, and inhibitory effects
33570-04-6 sc-201061
sc-201061B
sc-201061A
sc-201061C
10 mg
25 mg
50 mg
100 mg
$75.00
$142.00
$275.00
$420.00
3
(1)
(-)-Bicuculline methochloride
(−)-Bicuculline methochloride is a water-soluble GABAA antagonist
53552-05-9 sc-203528
sc-203528A
10 mg
50 mg
$109.00
$323.00
0
(0)
THIP hydrochloride
THIP hydrochloride is a GABAA receptor agonist and GABAC receptor antagonist
64603-91-4 sc-204342
50 mg
$149.00
0
(0)
beta-CCB
β-CCB is a benzodiazepine inverse agonist and putative endogenous ligand
84454-35-3 sc-204429
sc-204429A
10 mg
50 mg
$109.00
$460.00
0
(0)
DHEA
DHEA is a negative modulator of GABAA receptors
53-43-0 sc-202573
10 g
$101.00
1
(1)
2-Hydroxysaclofen
2-Hydroxysaclofen is a selective GABAB antagonist
117354-64-0 sc-202011
sc-202011A
2.5 mg
10 mg
$199.00
$180.00
0
(0)
CGP 46381
CGP 46381 is a selective GABAB receptor antagonist
123691-14-5 sc-361140
sc-361140A
10 mg
50 mg
$175.00
$739.00
0
(0)
SKF 89976A hydrochloride
SKF 89976A hydrochloride is a potent GABA uptake inhibitor
85375-85-5 sc-203266
sc-203266A
1 mg
10 mg
$30.00
$123.00
0
(0)
SCS
SCS is potent and selective partial inhibitor of β1-containing GABAA receptors
3232-36-8 sc-203375
50 mg
$105.00
0
(0)
Saclofen
Saclofen is a selective GABAB antagonist
125464-42-8 sc-203252
10 mg
$175.00
0
(0)
Etbicyphat
Etbicyphat is a synthetic, non-competitive GABA antagonist
1005-93-2 sc-294479
500 mg
$420.00
0
(0)
FrPbAII
FrPbAII is a GABA and glycine uptake inhibtor
sc-221630
5 mg
$450.00
0
(0)
Mebicyphat
Mebicyphat is a noncompetitive GABA antagonist
1449-89-4 sc-295376
500 mg
$395.00
0
(0)
CGP 36216
CGP 36216 is a GABAB selective antagonist
123691-29-2 sc-362724
sc-362724A
10 mg
50 mg
$155.00
$712.00
0
(0)
U 93631
U 93631 is a GABAA receptor antagonist
152273-12-6 sc-204364
sc-204364A
10 mg
50 mg
$169.00
$715.00
0
(0)
NNC 05-2090 hydrochloride
NNC 05-2090 hydrochloride is a GABA uptake inhibitor displaying selectivity for BGT-1 (mGAT-2) transporters
184845-43-0 sc-204131
sc-204131A
10 mg
50 mg
$214.00
$825.00
0
(0)
(S)-SNAP 5114
(S)-SNAP 5114 is a GABA uptake inhibitor that increases thalamic GABA levels
157604-55-2 sc-204257
sc-204257A
5 mg
25 mg
$115.00
$406.00
0
(0)
TB 21007
TB 21007 is a GABAA receptor inverse agonist
207306-50-1 sc-204322
sc-204322A
10 mg
50 mg
$169.00
$715.00
0
(0)
Vigabatrin
Vigabatrin is a selective GABA transaminase inhibitor
60643-86-9 sc-204382
sc-204382A
sc-204382B
sc-204382C
10 mg
50 mg
100 mg
1 g
$88.00
$359.00
$480.00
$700.00
2
(1)
Gabazine
Gabazine is a specific GABA receptor antagonist
105538-73-6 sc-211552
10 mg
$338.00
1
(0)
Furosemide-d5
Furosemide-d5 is an inhibitor of co-transport in the kidney
54-31-9 unlabeled sc-218550
sc-218550A
1 mg
10 mg
$280.00
$2,200.00
0
(0)
Cloflubicyne
Cloflubicyne is a potent non-competitive GABA antagonist
224790-70-9 sc-300382
1 mg
$260.00
0
(0)
DMCM hydrochloride
DMCM hydrochloride is a benzodiazepine inverse agonist
82499-00-1 sc-205295
sc-205295A
10 mg
50 mg
$190.00
$770.00
1
(0)
Droperidol
Droperidol is a D1DR and D2DR inhibitor
548-73-2 sc-211382
1 g
$110.00
0
(1)
ZK 93426 hydrochloride
ZK 93426 hydrochloride is a elective and competitive benzodiazepine receptor antagonist
89592-45-0 sc-203727
sc-203727A
10 mg
50 mg
$169.00
$630.00
0
(0)
Imidazole-4-acetic acid sodium salt
Imidazole-4-acetic acid sodium salt is a competitive antagonist at GABAC receptors
56368-58-2 sc-252900
sc-252900A
500 mg
1 g
$200.00
$300.00
0
(0)
Xli 093
Xli 093 is α5 subtype selective benzodiazepine/GABAA receptor antagonist
646066-59-3 sc-264494
5 mg
$134.00
0
(0)
β-Alanine
β-Alanine is an endogenous glycine agonist and GABA transporter inhibitor
107-95-9 sc-364682
sc-364682A
25 g
500 g
$30.00
$94.00
0
(0)

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