CGP 54626 hydrochloride (CAS 149184-21-4)
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CGP 54626 Hydrochloride is a selective and potent antagonist of the metabotropic glutamate receptor subtype 1 (mGluR1). It functions by binding to the receptor and inhibiting its activation by glutamate, thereby blocking the downstream signaling pathways. This chemical specifically targets the glutamate receptor in a competitive manner, preventing the binding of glutamate and subsequent activation of the receptor. By doing so, CGP 54626 Hydrochloride effectively modulates synaptic transmission and neuronal excitability mediated by mGluR1. This mechanism of action makes it a valuable tool for studying the physiological and pathological roles of mGluR1 in cellular and molecular processes. Additionally, its selective antagonistic properties allow for the investigation of the specific functions of mGluR1 without interference from other receptor subtypes. CGP 54626 Hydrochloride may play a significant role in understanding the molecular and cellular mechanisms involving mGluR1 in research and development applications.
CGP 54626 hydrochloride (CAS 149184-21-4) References
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Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
CGP 54626 hydrochloride, 10 mg | sc-361142 | 10 mg | $270.00 |