GABA Receptor Inhibitors
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Items 31 to 34 of 34 total
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| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
Droperidol | 548-73-2 | sc-211382 | 1 g | $190.00 | ||
Droperidol functions as a GABA receptor modulator, exhibiting unique allosteric properties that enhance receptor sensitivity to GABA. Its molecular structure facilitates specific interactions with the receptor's allosteric sites, promoting conformational changes that influence chloride ion permeability. This modulation alters synaptic transmission dynamics, with a distinctive profile of receptor activation and desensitization. The compound's kinetics reveal a complex interplay between binding affinity and receptor response, contributing to its nuanced effects on neural signaling pathways. | ||||||
DMCM hydrochloride | 82499-00-1 | sc-205295 sc-205295A | 10 mg 50 mg | $208.00 $832.00 | 2 | |
DMCM hydrochloride acts as a GABA receptor antagonist, uniquely disrupting the receptor's normal function. Its molecular interactions involve competitive binding at the GABA site, leading to altered chloride ion flow and reduced inhibitory neurotransmission. This compound exhibits distinctive kinetics, characterized by rapid onset and a short duration of action, which influences synaptic plasticity. The resulting changes in neuronal excitability highlight its role in modulating central nervous system activity. | ||||||
Imidazole-4-acetic acid sodium salt | 56368-58-2 | sc-252900 sc-252900A | 500 mg 1 g | $214.00 $318.00 | ||
Imidazole-4-acetic acid sodium salt functions as a GABA receptor modulator, engaging in allosteric interactions that enhance receptor sensitivity. Its unique structure allows for specific binding to auxiliary sites, facilitating increased chloride ion conductance. The compound exhibits a gradual onset of action, promoting sustained effects on synaptic transmission. This modulation of receptor dynamics can influence neuronal signaling pathways, contributing to the fine-tuning of excitatory and inhibitory balance in neural circuits. | ||||||
Xli 093 | 646066-59-3 | sc-264494 | 5 mg | $134.00 | ||
Xli 093 acts as a GABA receptor modulator, characterized by its ability to selectively bind to distinct allosteric sites, thereby altering receptor conformation. This interaction promotes enhanced chloride ion influx, leading to a pronounced effect on neuronal excitability. The compound exhibits unique reaction kinetics, with a rapid onset followed by a prolonged modulation of synaptic activity, influencing neurotransmitter release and receptor desensitization in neural networks. | ||||||