mGluR-4 Inhibitors
SEE ALSO...
| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
MAP4 | 157381-42-5 | sc-202221 | 5 mg | $40.00 | ||
MAP4 serves as a selective modulator of mGluR-4, exhibiting unique binding dynamics that promote receptor dimerization and allosteric modulation. Its structural conformation allows for specific hydrogen bonding and hydrophobic interactions, influencing downstream signaling cascades. The compound's kinetic profile reveals a slow dissociation rate, enhancing receptor activation duration. This behavior can lead to nuanced alterations in neurotransmitter release and synaptic efficacy, highlighting its role in fine-tuning neural communication. | ||||||
MSX-3 | 261717-23-1 | sc-255310 sc-255310A | 5 mg 25 mg | $233.00 $930.00 | ||
MSX-3 is a selective antagonist of mGluR-4 that has been used in research to investigate the effects of blocking mGluR-4 activity. | ||||||
(RS)-CPPG | 183364-82-1 | sc-203448 sc-203448A | 5 mg 25 mg | $416.00 $1248.00 | 1 | |
(RS)-CPPG acts as a selective modulator of mGluR-4, characterized by its ability to stabilize receptor conformations through specific electrostatic interactions. Its unique molecular architecture facilitates distinct allosteric effects, promoting enhanced receptor sensitivity to endogenous ligands. The compound exhibits a favorable binding affinity, leading to prolonged engagement with the receptor, which can subtly influence intracellular signaling pathways and neuronal excitability. | ||||||
UBP1112 | 339526-74-8 | sc-204368 sc-204368A | 10 mg 50 mg | $686.00 $1509.00 | 2 | |
UBP1112 serves as a selective modulator of mGluR-4, distinguished by its capacity to induce conformational changes in the receptor through targeted hydrophobic interactions. This compound's unique structural features enable it to selectively enhance receptor activity, thereby fine-tuning downstream signaling cascades. Its kinetic profile suggests rapid association and dissociation rates, allowing for dynamic modulation of receptor function in response to varying cellular conditions. | ||||||
MMPEP | 823198-78-3 | sc-215392 | 10 mg | $344.00 | ||
MPEP is another compound that acts as an antagonist of mGluR-It has been used in research studies to examine the role of mGluR-4 in various neural processes. | ||||||
MTPG | 169209-66-9 | sc-204106 sc-204106A | 5 mg 50 mg | $119.00 $709.00 | ||
MTPG acts as a selective modulator of mGluR-4, characterized by its ability to stabilize receptor dimers through specific electrostatic interactions. This compound exhibits a unique binding affinity that promotes allosteric modulation, influencing the receptor's conformational landscape. Its distinct kinetic behavior, marked by prolonged receptor engagement, facilitates sustained signaling pathways, thereby impacting cellular responses in a nuanced manner. | ||||||
ACPT-II | 195209-04-2 | sc-361100 sc-361100A | 10 mg 50 mg | $179.00 $739.00 | ||
ACPT-II serves as a selective modulator of mGluR-4, distinguished by its capacity to induce conformational changes in the receptor through unique hydrophobic interactions. This compound demonstrates a remarkable ability to enhance receptor desensitization, altering downstream signaling cascades. Its reaction kinetics reveal a rapid onset of action, coupled with a gradual dissociation profile, allowing for fine-tuned regulation of synaptic transmission and neuronal excitability. | ||||||
(RS)-MSPG | 169209-64-7 | sc-203247 sc-203247A | 5 mg 10 mg | $48.00 $201.00 | ||
(RS)-MSPG acts as a selective modulator of mGluR-4, characterized by its ability to stabilize receptor dimers through specific electrostatic interactions. This compound influences receptor activity by promoting allosteric modulation, which fine-tunes the receptor's response to glutamate. Its unique binding affinity leads to altered intracellular calcium signaling, impacting various neuronal pathways. The compound exhibits a distinct pharmacokinetic profile, facilitating prolonged receptor engagement. | ||||||