Estrogen Receptor Activators
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Items 1 to 10 of 13 total
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| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
Daidzein | 486-66-8 | sc-24001 sc-24001A sc-24001B | 100 mg 500 mg 5 g | $25.00 $75.00 $150.00 | 32 | |
Daidzein functions as a selective estrogen receptor modulator, engaging with estrogen receptors through specific hydrogen bonding and hydrophobic interactions. Its unique structure allows for differential activation of receptor subtypes, influencing gene expression pathways. The compound's conformational flexibility enhances its binding affinity, while its ability to stabilize receptor-ligand complexes can modulate downstream signaling cascades. This nuanced interaction profile contributes to its distinct biological effects. | ||||||
DHEA | 53-43-0 | sc-202573 | 10 g | $109.00 | 3 | |
DHEA acts as a modulator of estrogen receptors, exhibiting a unique ability to influence receptor conformation through specific hydrophobic and electrostatic interactions. Its structural characteristics allow it to selectively engage with various receptor subtypes, leading to differential activation of signaling pathways. The compound's dynamic nature facilitates rapid binding and dissociation kinetics, enabling it to fine-tune gene expression and cellular responses in a context-dependent manner. | ||||||
Tamoxifen Citrate | 54965-24-1 | sc-203288 | 100 mg | $81.00 | 12 | |
Tamoxifen Citrate functions as a selective estrogen receptor modulator, characterized by its ability to bind to estrogen receptors with high affinity. Its unique structure allows for distinct interactions with receptor domains, influencing conformational changes that alter downstream signaling. The compound exhibits a notable capacity for competitive inhibition, impacting the receptor's interaction with endogenous ligands. This selective binding profile contributes to its nuanced effects on gene regulation and cellular behavior. | ||||||
Diethylstilbestrol | 56-53-1 | sc-204720 sc-204720A sc-204720B sc-204720C sc-204720D | 1 g 5 g 25 g 50 g 100 g | $70.00 $281.00 $536.00 $1076.00 $2142.00 | 3 | |
Diethylstilbestrol acts as a potent estrogen receptor agonist, exhibiting a unique ability to stabilize receptor conformations that enhance transcriptional activity. Its synthetic structure allows for strong interactions with the ligand-binding domain, promoting dimerization and subsequent activation of estrogen-responsive genes. The compound's lipophilicity facilitates cellular uptake, while its prolonged half-life leads to sustained receptor engagement, influencing various signaling pathways and gene expression profiles. | ||||||
Raloxifene 4′-Glucuronide | 182507-22-8 | sc-222242 sc-222242A sc-222242B sc-222242C | 1 mg 2 mg 5 mg 10 mg | $403.00 $668.00 $1637.00 $2861.00 | 2 | |
Raloxifene 4'-Glucuronide functions as a selective estrogen receptor modulator, exhibiting distinct binding affinities that influence receptor conformation and activity. Its glucuronidation enhances solubility and alters pharmacokinetics, allowing for differential tissue distribution. The compound's unique interactions with the estrogen receptor can modulate downstream signaling cascades, impacting gene regulation. Additionally, its stability in biological systems contributes to its nuanced effects on receptor-mediated pathways. | ||||||
α-Zearalanol | 26538-44-3 | sc-391045 | 5 mg | $263.00 | ||
α-Zearalanol acts as a potent estrogen receptor agonist, engaging in specific hydrogen bonding and hydrophobic interactions that stabilize receptor-ligand complexes. This compound influences receptor dimerization and translocation, thereby modulating gene expression through distinct signaling pathways. Its unique structural features allow for selective activation of estrogen-responsive genes, while its metabolic stability ensures prolonged receptor engagement, enhancing its biological efficacy. | ||||||
α-Estradiol | 57-91-0 | sc-204425 | 50 mg | $70.00 | 1 | |
α-Estradiol is a key estrogen receptor ligand that exhibits high affinity for estrogen receptors, facilitating conformational changes that enhance receptor activity. Its unique hydroxyl groups enable specific interactions with amino acid residues, promoting effective receptor dimerization. This compound also influences downstream signaling cascades, impacting cellular responses. Additionally, its lipophilic nature aids in membrane permeability, allowing for rapid cellular uptake and interaction with intracellular targets. | ||||||
4,4′-(Hexafluoroisopropylidene)diphenol | 1478-61-1 | sc-262203 sc-262203A | 50 g 250 g | $77.00 $250.00 | 3 | |
4,4'-(Hexafluoroisopropylidene)diphenol acts as a selective estrogen receptor modulator, engaging in unique hydrogen bonding and hydrophobic interactions with receptor sites. Its distinct fluorinated structure enhances binding affinity and stability, influencing receptor conformation and activity. The compound's electronic properties facilitate specific molecular interactions, potentially altering gene expression pathways. Its robust stability under various conditions allows for consistent performance in receptor-mediated processes. | ||||||
Estropipate | 7280-37-7 | sc-203946 | 50 mg | $107.00 | 1 | |
Estropipate functions as a selective estrogen receptor modulator, characterized by its ability to form specific ionic and hydrophobic interactions with estrogen receptors. Its unique structural features promote a conformational change in the receptor, enhancing its activation potential. The compound's dynamic solubility and stability in diverse environments contribute to its effective engagement in cellular signaling pathways, influencing downstream biological responses. | ||||||
Triadimenol | 55219-65-3 | sc-205871 sc-205871A | 10 g 25 g | $116.00 $237.00 | ||
Triadimenol acts as a selective estrogen receptor modulator, exhibiting unique binding affinities that facilitate distinct conformational changes in the receptor. Its molecular structure allows for specific hydrogen bonding and hydrophobic interactions, which enhance receptor activation. The compound's kinetic profile reveals a rapid association and dissociation with the receptor, influencing gene expression and cellular responses. Additionally, its solubility characteristics enable effective distribution within biological systems. | ||||||