CYPOR Inhibitors
Items 1 to 10 of 12 total
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| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
7-Ethoxyresorufin | 5725-91-7 | sc-200606 sc-200606A | 2 mg 10 mg | $138.00 $270.00 | 6 | |
7-Ethoxyresorufin serves as a selective substrate for cytochrome P450 enzymes, particularly CYP1A1. Its unique structure allows for efficient electron transfer during metabolic reactions, leading to the formation of fluorescent metabolites. The compound exhibits distinct reaction kinetics, with a rapid conversion rate that highlights its sensitivity to enzyme activity. Additionally, its hydrophilic and lipophilic balance enhances membrane permeability, influencing its bioavailability and interaction with various biological systems. | ||||||
Amodiaquine | 86-42-0 | sc-207282 | 10 mg | $342.00 | 1 | |
Amodiaquine is a direct inhibitor of CYPOR, specifically interfering with its electron transfer function. It disrupts the electron transport chain by binding to CYPOR and preventing the efficient transfer of electrons from NADPH to cytochrome P450 enzymes. | ||||||
Fluconazole | 86386-73-4 | sc-205698 sc-205698A | 500 mg 1 g | $54.00 $84.00 | 14 | |
Fluconazole is a direct inhibitor of CYPOR, acting on its electron transfer function. By binding to CYPOR, it interferes with the transfer of electrons from NADPH to cytochrome P450 enzymes, particularly those involved in the synthesis of sterols. | ||||||
Fenofibrate | 49562-28-9 | sc-204751 | 5 g | $41.00 | 9 | |
Fenofibrate is a direct inhibitor of CYPOR, targeting its electron transfer function. It interferes with the transfer of electrons from NADPH to cytochrome P450 enzymes, leading to a reduction in their enzymatic activity. | ||||||
Erythromycin | 114-07-8 | sc-204742 sc-204742A sc-204742B sc-204742C | 5 g 25 g 100 g 1 kg | $57.00 $245.00 $831.00 $1331.00 | 4 | |
Erythromycin is a direct inhibitor of CYPOR, specifically affecting its electron transfer activity. By binding to CYPOR, it disrupts the flow of electrons from NADPH to cytochrome P450 enzymes, leading to a decrease in their catalytic function. | ||||||
Clotrimazole | 23593-75-1 | sc-3583 sc-3583A | 100 mg 1 g | $42.00 $57.00 | 6 | |
Clotrimazole is a direct inhibitor of CYPOR, acting on its electron transfer function. It interferes with the transfer of electrons from NADPH to cytochrome P450 enzymes, particularly those involved in the synthesis of sterols. | ||||||
17-AAG | 75747-14-7 | sc-200641 sc-200641A | 1 mg 5 mg | $67.00 $156.00 | 16 | |
17-AAG is a direct inhibitor of CYPOR, targeting its electron transfer function. It disrupts the flow of electrons from NADPH to cytochrome P450 enzymes, leading to a decrease in their catalytic activity. | ||||||
Trimethoprim | 738-70-5 | sc-203302 sc-203302A sc-203302B sc-203302C sc-203302D | 5 g 25 g 250 g 1 kg 5 kg | $67.00 $161.00 $255.00 $721.00 $3401.00 | 4 | |
Trimethoprim is a direct inhibitor of CYPOR, specifically affecting its electron transfer activity. By binding to CYPOR, it disrupts the transfer of electrons from NADPH to cytochrome P450 enzymes, leading to a decrease in their enzymatic function. | ||||||
Tamoxifen | 10540-29-1 | sc-208414 | 2.5 g | $272.00 | 18 | |
Tamoxifen is a direct inhibitor of CYPOR, acting on its electron transfer function. It interferes with the transfer of electrons from NADPH to cytochrome P450 enzymes, particularly those involved in the metabolism of endogenous and exogenous compounds. | ||||||
Ketoconazole | 65277-42-1 | sc-200496 sc-200496A | 50 mg 500 mg | $63.00 $265.00 | 21 | |
Ketoconazole is a direct inhibitor of CYPOR, targeting its electron transfer function. It disrupts the flow of electrons from NADPH to cytochrome P450 enzymes, leading to a decrease in their catalytic activity. | ||||||