Ser/Thr Protein Kinase Inhibitors
Items 251 to 260 of 284 total
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| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
3-Methyl 7-Azaoxindole | 1330055-85-0 | sc-482877 | 50 mg | $380.00 | ||
3-Methyl 7-Azaoxindole functions as a Ser/Thr protein kinase inhibitor, characterized by its ability to engage in specific hydrogen bonding and hydrophobic interactions within the kinase domain. This compound stabilizes inactive conformations of the enzyme, effectively blocking substrate phosphorylation. Its unique structural features facilitate selective binding, influencing downstream signaling cascades and providing a deeper understanding of kinase regulation in cellular processes. | ||||||
Pseudohypericin | 55954-61-5 | sc-202777 sc-202777A | 1 mg 5 mg | $156.00 $599.00 | ||
Pseudohypericin acts as a Ser/Thr protein kinase modulator, exhibiting unique binding dynamics that enhance its interaction with the kinase domain. Its distinct molecular architecture allows for the formation of critical electrostatic interactions, which can alter the enzyme's conformational states. This compound influences reaction kinetics by stabilizing transition states, thereby affecting substrate affinity and phosphorylation rates, ultimately impacting various signaling pathways within the cell. | ||||||
β-Glycerophosphate disodium salt | 819-83-0 | sc-220452 sc-220452A sc-220452B sc-220452C sc-220452D sc-220452E | 25 g 100 g 500 g 1 kg 3 kg 6 kg | $63.00 $119.00 $442.00 $738.00 $2091.00 $3652.00 | 43 | |
β-Glycerophosphate disodium salt serves as a potent modulator of Ser/Thr protein kinases, characterized by its ability to mimic phosphate groups in cellular signaling. Its unique structural features facilitate specific interactions with kinase active sites, promoting conformational changes that enhance enzymatic activity. This compound also influences the phosphorylation cascade by altering substrate recognition and binding dynamics, thereby playing a crucial role in regulating cellular processes and signal transduction pathways. | ||||||
3-(2,7-Dimethoxy-acridin-9-ylsulfanyl)-propylamine dihydrochloride | 184582-62-5 (free base) | sc-396704 sc-396704A | 5 mg 25 mg | $80.00 $341.00 | ||
3-(2,7-Dimethoxy-acridin-9-ylsulfanyl)-propylamine dihydrochloride exhibits a distinctive mechanism of action as a Ser/Thr protein kinase modulator. Its unique acridine scaffold allows for selective interactions with the ATP-binding pocket, promoting conformational changes that hinder substrate access. This compound's ability to disrupt kinase dimerization and alter allosteric sites enhances its specificity, providing insights into the regulatory mechanisms of cellular signaling pathways. | ||||||
Elbfluorene | sc-221585 sc-221585A | 1 mg 5 mg | $200.00 $400.00 | |||
Elbfluorene is a selective modulator of Ser/Thr protein kinases, characterized by its unique ability to engage in specific hydrogen bonding interactions that stabilize the kinase's inactive state. This compound influences the conformational dynamics of the enzyme, leading to altered phosphorylation rates. Its distinct molecular architecture facilitates unique interactions with substrate binding sites, thereby affecting signal transduction pathways and cellular regulatory networks. | ||||||
Guanosine-3′,5′-cyclic Monophosphothioate, Sp-Isomer sodium salt | 86562-10-9 | sc-203065 sc-203065A | 500 µg 1 mg | $200.00 $400.00 | ||
Guanosine-3',5'-cyclic Monophosphothioate, Sp-Isomer sodium salt acts as a potent modulator of Ser/Thr protein kinases, exhibiting a unique affinity for the enzyme's active site. Its thioate modification enhances binding stability and alters the enzyme's catalytic efficiency. This compound can influence the phosphorylation cascade by selectively disrupting or enhancing interactions with downstream substrates, thereby modulating critical cellular signaling pathways and regulatory mechanisms. | ||||||
SBI-0206965 | 1884220-36-3 | sc-507431 | 10 mg | $124.00 | ||
(R)-2-((9-Isopropyl-6-((3-(pyridin-2-yl)phenyl)-amino)-9H-purin-2-yl)amino)butan-1-ol | 1056016-06-8 | sc-296248 sc-296248A | 50 mg 100 mg | $800.00 $1400.00 | ||
(R)-2-((9-Isopropyl-6-((3-(pyridin-2-yl)phenyl)-amino)-9H-purin-2-yl)amino)butan-1-ol serves as a selective inhibitor of Ser/Thr protein kinases, showcasing a unique structural conformation that facilitates specific interactions with the kinase domain. Its intricate design allows for tailored binding, influencing the enzyme's conformational dynamics and phosphorylation activity. This compound can modulate substrate recognition and alter downstream signaling events, impacting cellular responses. | ||||||
CR8, (S)-Isomer | 1084893-56-0 | sc-311307 | 5 mg | $201.00 | ||
CR8, the (S)-isomer, exhibits a distinctive binding affinity for Ser/Thr protein kinases, characterized by its unique stereochemistry that enhances interaction with the ATP-binding site. This compound's specific molecular architecture promotes selective inhibition, effectively disrupting kinase-mediated phosphorylation cascades. Its kinetic profile reveals a nuanced modulation of enzyme activity, influencing substrate specificity and downstream signaling pathways, thereby altering cellular regulatory mechanisms. | ||||||
TCS 21311 | 1260181-14-3 | sc-362804 sc-362804A | 10 mg 50 mg | $270.00 $1077.00 | ||
TCS 21311 is a selective inhibitor of Ser/Thr protein kinases, distinguished by its unique structural motifs that facilitate precise interactions with the enzyme's active site. This compound exhibits a remarkable ability to modulate phosphorylation events, impacting key signaling pathways. Its reaction kinetics suggest a competitive inhibition mechanism, allowing for fine-tuning of kinase activity and influencing cellular processes through altered substrate interactions and regulatory feedback loops. | ||||||