NMDA zeta 1 Inhibitors
| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
TCS 46b | 302799-86-6 | sc-204328 sc-204328A | 10 mg 50 mg | $149.00 $630.00 | ||
TCS 46b acts as a selective NMDA zeta 1 modulator, characterized by its ability to engage in specific hydrogen bonding interactions with receptor sites. This compound influences ion channel permeability, leading to altered excitatory neurotransmission. Its unique steric configuration enhances binding affinity, while its lipophilic characteristics facilitate membrane partitioning, affecting its distribution and reactivity in various biochemical environments. The compound's kinetic behavior is marked by rapid association and dissociation rates, underscoring its dynamic role in synaptic modulation. | ||||||
Memantine hydrochloride | 41100-52-1 | sc-203628 | 50 mg | $68.00 | 4 | |
Memantine is another NMDA receptor antagonist. It preferentially blocks excessive NMDA receptor activity without disrupting normal activity, thereby indirectly inhibiting NMDAζ1. | ||||||
Dextromethorphan | 125-71-3 | sc-278927 sc-278927A sc-278927B | 10 g 100 g 500 g | $174.00 $1133.00 $5106.00 | 3 | |
Dextromethorphan acts as an NMDA receptor antagonist. It can inhibit NMDAζ1 by interfering with the receptor's normal function in synaptic transmission. | ||||||
Ifenprodil hemitartrate | 23210-58-4 | sc-203601B sc-203601 sc-203601A | 5 mg 10 mg 50 mg | $39.00 $61.00 $142.00 | ||
Ifenprodil selectively inhibits certain subtypes of NMDA receptors. It can indirectly inhibit NMDAζ1 by modulating receptor activity, particularly in receptors containing the NR2B subunit. | ||||||
1-Adamantylamine | 768-94-5 | sc-251475 sc-251475A | 1 g 25 g | $38.00 $144.00 | ||
Amantadine has NMDA receptor antagonist properties. It can inhibit NMDAζ1 by altering the receptor's function in neural transmission and plasticity. | ||||||
Felbamate | 25451-15-4 | sc-203579 sc-203579A | 10 mg 50 mg | $101.00 $373.00 | ||
Felbamate has been shown to modulate NMDA receptor activity. It can indirectly inhibit NMDAζ1 by affecting the receptor's function in synaptic transmission. | ||||||
Ifenprodil Tartrate Salt | 23210-56-2 | sc-295173 sc-295173A | 5 mg 10 mg | $55.00 $71.00 | ||
Ifenprodil Tartrate Salt functions as a selective NMDA zeta 1 antagonist, exhibiting unique electrostatic interactions that stabilize its binding to receptor sites. This compound alters calcium ion influx, impacting synaptic plasticity. Its distinct conformational flexibility allows for effective competition with endogenous ligands, while its hydrophilic nature influences solubility and diffusion across cellular membranes. The compound's reaction kinetics reveal a notable balance between affinity and dissociation, contributing to its nuanced role in neurophysiological processes. | ||||||
Riluzole | 1744-22-5 | sc-201081 sc-201081A sc-201081B sc-201081C | 20 mg 100 mg 1 g 25 g | $20.00 $189.00 $209.00 $311.00 | 1 | |
Riluzole modulates glutamatergic neurotransmission and can inhibit NMDA receptors. It indirectly inhibits NMDAζ1 by affecting synaptic transmission mediated by these receptors. | ||||||