GAK Inhibitors
Items 1 to 10 of 13 total
Display:
| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
SB 203580 | 152121-47-6 | sc-3533 sc-3533A | 1 mg 5 mg | $90.00 $349.00 | 284 | |
SB 203580 is a selective inhibitor that targets the p38 mitogen-activated protein kinase (MAPK) pathway, exhibiting unique molecular interactions that modulate cellular stress responses. Its structure allows for specific binding to the ATP-binding site, altering phosphorylation dynamics and influencing downstream signaling cascades. The compound's hydrophobic regions enhance membrane permeability, affecting its distribution and interaction with various cellular compartments, thereby impacting cellular function. | ||||||
Alsterpaullone | 237430-03-4 | sc-202453 sc-202453A | 1 mg 5 mg | $68.00 $312.00 | 2 | |
Alsterpaullone is a cyclin-dependent kinase inhibitor that may inhibit GAK by affecting its association with cyclins. | ||||||
Roscovitine | 186692-46-6 | sc-24002 sc-24002A | 1 mg 5 mg | $94.00 $265.00 | 42 | |
Roscovitine targets various cyclin-dependent kinases and could impede GAK's kinase activity by competitive inhibition. | ||||||
Indirubin-3′-monoxime | 160807-49-8 | sc-202660 sc-202660A sc-202660B | 1 mg 5 mg 50 mg | $79.00 $321.00 $671.00 | 1 | |
This compound is a CDK inhibitor that might also inhibit GAK due to its role in cell cycle regulation. | ||||||
Hesperadin | 422513-13-1 | sc-490384 | 10 mg | $304.00 | ||
Hesperadin is an Aurora kinase inhibitor, which could indirectly affect GAK by altering cell cycle progression. | ||||||
SP600125 | 129-56-6 | sc-200635 sc-200635A | 10 mg 50 mg | $40.00 $150.00 | 257 | |
As a JNK inhibitor, SP600125 can modulate stress-response pathways potentially related to GAK's functions. | ||||||
5-Iodotubercidin | 24386-93-4 | sc-3531 sc-3531A | 1 mg 5 mg | $153.00 $464.00 | 20 | |
This adenosine analog inhibits various kinases and could non-selectively inhibit GAK's ATP-binding site. | ||||||
Harmine | 442-51-3 | sc-202644 sc-202644A sc-202644B sc-202644C sc-202644D sc-202644E sc-202644F | 250 mg 500 mg 1 g 10 g 50 g 100 g 500 g | $53.00 $104.00 $126.00 $551.00 $1467.00 $2611.00 $11455.00 | 2 | |
Harmine is a DYRK inhibitor that might affect GAK activity through overlaps in substrate specificity or pathway interaction. | ||||||
Purvalanol A | 212844-53-6 | sc-224244 sc-224244A | 1 mg 5 mg | $72.00 $297.00 | 4 | |
Purvalanol A is a CDK inhibitor that could also inhibit GAK, impacting cell cycle and transcription regulation. | ||||||
Dinaciclib | 779353-01-4 | sc-364483 sc-364483A | 5 mg 25 mg | $247.00 $888.00 | 1 | |
Dinaciclib strongly inhibits CDKs and might inhibit GAK, potentially affecting downstream signaling. | ||||||