ERR gamma Activators
Items 1 to 10 of 17 total
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| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
Fenofibrate | 49562-28-9 | sc-204751 | 5 g | $41.00 | 9 | |
Fenofibrate, a PPARα agonist, is known to upregulate the expression of ERRγ. By activating PPARα, fenofibrate increases the expression of PGC-1α, a transcriptional coactivator, which directly interacts with and enhances the transcriptional activity of ERRγ. | ||||||
DY131 | 95167-41-2 | sc-203571 sc-203571A | 10 mg 50 mg | $132.00 $520.00 | 1 | |
DY131 is a selective modulator of ERR gamma, distinguished by its unique ability to form stable complexes through π-π stacking and van der Waals interactions. This compound influences metabolic pathways by altering transcriptional activity, effectively reshaping gene expression profiles. Its structural design allows for precise molecular docking, enhancing its specificity and efficacy in targeting ERR gamma, thereby providing a deeper understanding of its regulatory mechanisms in cellular processes. | ||||||
GSK 4716 | 101574-65-6 | sc-203986 sc-203986A | 10 mg 50 mg | $71.00 $285.00 | ||
A synthetic agonist of ERRγ, known to enhance its transcriptional activity. | ||||||
GW 3965 hydrochloride | 405911-17-3 | sc-224011 sc-224011A sc-224011B | 5 mg 25 mg 1 g | $140.00 $483.00 $3121.00 | ||
GW3965 is a potent and selective agonist of liver X receptor (LXR), which is known to upregulate the expression of ERRγ. By activating LXR, GW3965 induces the expression of SREBP-1c, a transcription factor, which then enhances the transcriptional activity of ERRγ. | ||||||
Rosiglitazone | 122320-73-4 | sc-202795 sc-202795A sc-202795C sc-202795D sc-202795B | 25 mg 100 mg 500 mg 1 g 5 g | $120.00 $326.00 $634.00 $947.00 $1259.00 | 38 | |
Rosiglitazone is a PPARγ agonist that stimulates PGC-1α, a coactivator of ERRγ. The enhanced PGC-1α activity leads to upregulation of ERRγ transcriptional activity. | ||||||
Pioglitazone | 111025-46-8 | sc-202289 sc-202289A | 1 mg 5 mg | $55.00 $125.00 | 13 | |
Pioglitazone, a PPARγ agonist, enhances PGC-1α activity which in turn upregulates ERRγ transcriptional activity. | ||||||
AICAR | 2627-69-2 | sc-200659 sc-200659A sc-200659B | 50 mg 250 mg 1 g | $65.00 $280.00 $400.00 | 48 | |
AICAR is an activator of AMP-activated protein kinase (AMPK). Activation of AMPK leads to increased PGC-1α activity, which can enhance the transcriptional activity of ERRγ. | ||||||
Nobiletin | 478-01-3 | sc-202733 | 10 mg | $189.00 | 2 | |
A natural flavonoid that has been reported to function as an ERRγ agonist, affecting energy metabolism. | ||||||
Metformin | 657-24-9 | sc-507370 | 10 mg | $79.00 | 2 | |
Metformin is an AMPK activator. By activating AMPK, it promotes PGC-1α activity which then enhances the transcriptional function of ERRγ. | ||||||
Bisphenol A | 80-05-7 | sc-391751 sc-391751A | 100 mg 10 g | $300.00 $490.00 | 5 | |
A controversial environmental estrogen that has shown the ability to activate ERRγ in certain studies. | ||||||