SEE ALSO...
| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
ICI 182,780 | 129453-61-8 | sc-203435 sc-203435A | 1 mg 10 mg | $83.00 $187.00 | 34 | |
ICI 182,780 is a selective estrogen receptor degrader (SERD) that works by binding to the estrogen receptor and promoting its degradation, leading to a decrease in estrogen signaling. | ||||||
Anastrozole | 120511-73-1 | sc-217647 | 10 mg | $92.00 | 1 | |
Anastrozole is an aromatase inhibitor that reduces the production of estrogen by inhibiting the aromatase enzyme. | ||||||
Letrozole | 112809-51-5 | sc-204791 sc-204791A | 25 mg 50 mg | $87.00 $147.00 | 5 | |
Letrozole is another aromatase inhibitor that works similarly to anastrozole by reducing estrogen production. | ||||||
Exemestane | 107868-30-4 | sc-203045 sc-203045A | 25 mg 100 mg | $134.00 $411.00 | ||
Exemestane is an aromatase inhibitor that irreversibly binds to the aromatase enzyme, blocking estrogen synthesis. | ||||||
Tamoxifen | 10540-29-1 | sc-208414 | 2.5 g | $272.00 | 18 | |
Although not a direct ESR1 inhibitor, tamoxifen is a selective estrogen receptor modulator (SERM) that competes with estrogen for binding to the estrogen receptor, effectively blocking estrogen's actions. | ||||||
Raloxifene | 84449-90-1 | sc-476458 | 1 g | $802.00 | 3 | |
Similar to tamoxifen, raloxifene is a SERM that has antiestrogenic effects on breast tissue. | ||||||