GSK Inhibitors

Glycogen synthase kinase 3, or GSK-3, is a serine/threonine, proline-directed kinase involved in a diverse array of signaling pathways, including glycogen synthesis and cellular adhesion, and has been implicated in Alzheimer's disease. Biochemicals that inhibit GSK have many applications in biochemical and physiological research. Click on the product name to view detailed information such as the chemical structure and specific chemical properties for each of our GSK Inhibitors. In stock GSK Inhibitors are available for immediate shipping.

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PRODUCT NAME/Application CAS Catalog # QUANTITY Price Citations RATING
Ro 31-8220
Ro 31-8220 is a cell-permeable PKC inhibitor that has been shown to be selective for PKC over CaM kinase II and PKA
138489-18-6 sc-200619
sc-200619A
1 mg
5 mg
$81.00
$220.00
15
(1)
Kenpaullone
Kenpaullone is a Cdk and GKS-3 inhibitor
142273-20-9 sc-200643
sc-200643A
sc-200643B
sc-200643C
1 mg
5 mg
10 mg
25 mg
$59.00
$147.00
$222.00
$485.00
1
(1)
SB-216763
SB-216763 is a potent, selective and ATP-competitive inhibitor of GSK-3α and GSK-3β
280744-09-4 sc-200646
sc-200646A
1 mg
5 mg
$64.00
$189.00
18
(1)
Cdk1/5 Inhibitor
Cdk1/5 Inhibitor is a 3-amino substituted pyrazoloquinoxaline compound and selective inhibitor of Cdk1/Cdk5
40254-90-8 sc-202094
sc-202094A
sc-202094B
1 mg
5 mg
10 mg
$60.00
$200.00
$360.00
2
(1)
Valproic acid sodium salt
Valproic acid sodium salt is an HDAC inhibitor with anticancer, anti-inflammatory and neuroprotective effects
1069-66-5 sc-202378A
sc-202378
sc-202378B
sc-202378C
1 g
5 g
25 g
100 g
$20.00
$31.00
$120.00
$355.00
7
(1)
Bisindolylmaleimide I (GF 109203X)
Bisindolylmaleimide I (GF 109203X) is a highly selective inhibitor of all PKC isoforms and slight inhibitor of GSK-3
133052-90-1 sc-24003
sc-24003A
5 mg
1 mg
$195.00
$83.00
33
(1)
Bisindolylmaleimide I, HCl
Bisindolylmaleimide I, HCl is a water soluble inhibitor for all known isoforms of PKC
176504-36-2 sc-24004
1 mg
$139.00
13
(1)
4-Bromoindole
4-Bromoindole is a potential inhibitor of GSK-3
52488-36-5 sc-216790
100 mg
$205.00
0
(0)
Indole-3-acetamide
Indole-3-acetamide is a GSK-3β, VEGF, and JAK3 inhibitor
879-37-8 sc-255213
sc-255213A
1 g
5 g
$44.00
$198.00
1
(0)
GSK-3 Inhibitor XIII
GSK-3 Inhibitor XIII is an ATP-binding site inhibitor of GSK-3
404828-08-6 sc-203987
sc-203987A
1 mg
5 mg
$158.00
$462.00
1
(0)
BIP-135
BIP-135 is a GSK-3 inibitor with modest efficacy against PKC and PI3K
941575-71-9 sc-364435
sc-364435A
5 mg
25 mg
$105.00
$410.00
0
(0)
Ellagic Acid, Dihydrate
Ellagic Acid, Dihydrate is a CK2, Topo I and II, FGR, GSK, and PKA inhibitor
476-66-4 sc-202598
sc-202598A
sc-202598B
sc-202598C
500 mg
5 g
25 g
100 g
$50.00
$85.00
$229.00
$693.00
7
(1)
GSK-3 Inhibitor IX
GSK-3 Inhibitor IX is a cell-permeable, highly potent, selective, reversible, and ATP-competitive inhibitor of GSK-3α and GSK-3β.
667463-62-9 sc-202634
sc-202634A
sc-202634B
1 mg
10 mg
50 mg
$56.00
$180.00
$850.00
10
(1)
GSK-3beta Inhibitor VII
GSK-3β Inhibitor VII is a cell-permeable, and non-ATP competitive inhibitor of GSK-3β
99-73-0 sc-202635
5 mg
$129.00
0
(0)
GSK-3beta Inhibitor VIII
GSK-3β Inhibitor VIII is a potent, selective inhibitor of GSK-3β
487021-52-3 sc-202636
sc-202636A
5 mg
10 mg
$128.00
$144.00
4
(1)
Aloisine, RP106
Aloisine, RP106 is a selective, potent, ATP-competitive inhibitor of Cdc 2 (CDK1)/cyclin B, CDK5/p25, and GSK-3
496864-15-4 sc-202452
sc-202452A
1 mg
5 mg
$31.00
$139.00
0
(0)
Indirubin-3'-monoxime
Indirubin-3′-monoxime is A potent inhibitor of GSK-3β, Cdk1, and Cdk5
160807-49-8 sc-202660
sc-202660A
sc-202660B
1 mg
5 mg
50 mg
$75.00
$309.00
$645.00
1
(1)
(Methoxycarbonylmethyl)triphenylphosphonium bromide
(Methoxycarbonylmethyl)triphenylphosphonium bromide is a reactant for the synthesis of GSK-3 inhibitors using the Wittig reaction
1779-58-4 sc-228467
50 g
$67.00
0
(0)
Isogranulatimide
Isogranulatimide is cell-permeable alkaloid that acts as a potent and ATP-competitive inhibitor of Chk1
244148-46-7 sc-202667
1 mg
$700.00
0
(0)
GSK-3beta Inhibitor XI
GSK-3β Inhibitor XI is a potent and specific ATP-competitive inhibitor of GSK-3β
626604-39-5 sc-204770
1 mg
$224.00
4
(1)
SB-415286
SB-415286 is an ATP-competitive inhibitor of GSK3α and GSK-3β
264218-23-7 sc-204901
sc-204901A
1 mg
5 mg
$62.00
$140.00
4
(1)
GSK-3 Inhibitor IX, Control, MeBIO
GSK-3 Inhibitor IX, Control, MeBIO is a cell-permeable N-methylated kinase inactive analog of GSK-3 Inhibitor IX
710323-61-8 sc-221688
1 mg
$135.00
0
(1)
GSK-3 Inhibitor X
GSK-3 Inhibitor X is a selective GSK-3α/β inhibitor
740841-15-0 sc-221689
5 mg
$140.00
4
(1)
5-Bromoindole
5-Bromoindole is a potential inhibitor of GSK-3
10075-50-0 sc-256902
5 g
$28.00
0
(0)
GSK-3 Inhibitor XVI
GSK-3 Inhibitor XVI is a compound that acts as potent, ATP-competitive & highly selective GSK-3 inhibitor.
252917-06-9 sc-221691
sc-221691A
5 mg
25 mg
$140.00
$500.00
3
(1)
GSK-3β Inhibitor I
GSK-3β Inhibitor I is a thiadiazolidinone analog that acts as a highly selective, non-ATP competitive inhibitor of GSK-3β
327036-89-5 sc-221692
sc-221692A
5 mg
25 mg
$179.00
$282.00
4
(0)
GSK-3beta Inhibitor VI
GSK-3β Inhibitor VI is a cell-permeable, irreversible, and non-ATP competitive inhibitor of GSK-3β
62673-69-2 sc-221693
5 mg
$220.00
1
(0)
GSK-3beta Inhibitor XII, TWS119
GSK-3β Inhibitor XII, TWS119 is a cell-permeable agent shown to act as a potent inhibitor of GSK-3β
601514-19-6 sc-221694
sc-221694A
1 mg
5 mg
$55.00
$150.00
10
(1)
Indirubin-3prime-monoxime-5-sulphonic Acid
Indirubin-3′-monoxime-5-sulphonic Acid is an inhibitor of GSK-3β, Cdc2 (Cdk1) and Cdk5.
331467-05-1 sc-221753
1 mg
$179.00
1
(0)
5-Iodo-Indirubin-3prime-monoxime
5-Iodo-Indirubin-3′-monoxime is an inhibitor of GSK-3β, CDK-1, and CDK-5
sc-221754
1 mg
$104.00
0
(0)
GSK-3 Inhibitor II
GSK-3 Inhibitor II is A potent GSK-3β inhibitor
478482-75-6 sc-24020
sc-24020A
5 mg
25 mg
$80.00
$290.00
10
(1)
1-Azakenpaullone
1-Azakenpaullone is a Kenpaullone analog and an inhibitor of GSK-3
676596-65-9 sc-358615
1 mg
$96.00
0
(0)
TCS 2002
TCS 2002 is a cell-permeable inhibitor of GSK-3β
1005201-24-0 sc-359020
sc-359020A
10 mg
50 mg
$175.00
$739.00
0
(0)
3F8
3F8 is a selective and potent GSK-3β inhibitor
159109-11-2 sc-361080
sc-361080A
10 mg
50 mg
$179.00
$756.00
1
(0)
TCS 21311
TCS 21311 is a potent inhibitor of JAK3
1260181-14-3 sc-362804
sc-362804A
10 mg
50 mg
$255.00
$1,030.00
0
(0)
A 1070722
A 1070722 is an inhibitor of GSK-3α and GSK-3β with a Ki = 0.6 nM respectively
1384424-80-9 sc-364392
sc-364392A
10 mg
50 mg
$131.00
$709.00
0
(0)