Date published: 2026-5-27

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4-Bromoindole (CAS 52488-36-5)

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Application:
4-Bromoindole is a potential inhibitor of GSK-3
CAS Number:
52488-36-5
Molecular Weight:
196.04
Molecular Formula:
C8H6BrN
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.

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4-Bromoindole is a potential inhibitor of GSK-3.


4-Bromoindole (CAS 52488-36-5) References

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  2. GSK-3-selective inhibitors derived from Tyrian purple indirubins.  |  Meijer, L., et al. 2003. Chem Biol. 10: 1255-66. PMID: 14700633
  3. A new synthesis of lysergic acid.  |  Hendrickson, JB. and Wang, J. 2004. Org Lett. 6: 3-5. PMID: 14703336
  4. Protein kinase inhibitors: insights into drug design from structure.  |  Noble, ME., et al. 2004. Science. 303: 1800-5. PMID: 15031492
  5. Glycogen synthase kinase-3beta mediates convergence of protection signaling to inhibit the mitochondrial permeability transition pore.  |  Juhaszova, M., et al. 2004. J Clin Invest. 113: 1535-49. PMID: 15173880
  6. Synthetic Studies on the Ambiguine Family of Alkaloids: Construction of the ABCD Ring System.  |  Rafferty, RJ. and Williams, RM. 2011. Tetrahedron Lett. 52: 2037-2040. PMID: 21516192
  7. [Development of unprotected syntheses in aqueous media].  |  Yokoyama, Y. 2013. Yakugaku Zasshi. 133: 249-68. PMID: 23370521
  8. Asymmetric formal synthesis of (+)-cycloclavine.  |  Chen, JQ., et al. 2017. Chem Commun (Camb). 53: 12902-12905. PMID: 29110004
  9. A Ten-Step Total Synthesis of Speradine C.  |  Liu, H., et al. 2019. Angew Chem Int Ed Engl. 58: 6362-6365. PMID: 30882976
  10. Enantioselective Formal Synthesis of (+)-Cycloclavine and Total Synthesis of (+)-5-epi-Cycloclavine.  |  Wang, W., et al. 2019. Org Lett. 21: 6603-6607. PMID: 31411477

Ordering Information

Product NameCatalog #UNITPriceQtyFAVORITES

4-Bromoindole, 100 mg

sc-216790
100 mg
$205.00