mGluR-4 Activators
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Items 11 to 15 of 15 total
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| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
TCN 238 | 125404-04-8 | sc-362803 sc-362803A | 10 mg 50 mg | $155.00 $620.00 | ||
TCN 238 is a potent modulator of mGluR-4, characterized by its ability to stabilize receptor conformations that favor specific signaling pathways. This compound exhibits unique interactions with the receptor's binding sites, leading to enhanced selectivity in downstream signaling events. Its kinetic behavior suggests a rapid onset of action, allowing for precise modulation of receptor activity. The structural attributes of TCN 238 facilitate its role in influencing synaptic plasticity through targeted receptor engagement. | ||||||
VU 0361737 | 1161205-04-4 | sc-301976 sc-301976A | 10 mg 50 mg | $115.00 $440.00 | ||
VU 0361737 is a selective allosteric modulator of mGluR-4, distinguished by its capacity to induce conformational changes that enhance receptor functionality. This compound engages with distinct allosteric sites, promoting unique signaling cascades that differ from orthosteric ligands. Its interaction profile suggests a nuanced influence on receptor dynamics, potentially altering desensitization rates and enhancing signal transduction efficiency, thereby contributing to intricate neural network modulation. | ||||||
VU 0364439 | 1246086-78-1 | sc-364720 sc-364720A | 10 mg 50 mg | $159.00 $795.00 | ||
VU 0364439 acts as a selective modulator of mGluR-4, characterized by its ability to stabilize specific receptor conformations. This compound selectively binds to allosteric sites, facilitating unique interactions that fine-tune receptor activity. Its kinetic profile indicates a rapid onset of action, influencing downstream signaling pathways and receptor phosphorylation states. The compound's distinct binding dynamics may also impact receptor trafficking and localization, contributing to its regulatory role in synaptic plasticity. | ||||||
MPEP hydrochloride | 96206-92-7 | sc-279454A sc-279454 | 10 mg 50 mg | $136.00 $520.00 | ||
MPEP hydrochloride is a selective allosteric modulator of mGluR-4, known for its unique ability to enhance receptor signaling through specific conformational changes. It engages with distinct binding sites, promoting nuanced interactions that alter receptor dynamics. The compound exhibits a favorable kinetic profile, allowing for swift modulation of intracellular pathways. Its influence on receptor desensitization and internalization may play a critical role in synaptic regulation and neuronal communication. | ||||||
L-γ-Carboxyglutamic acid | 53861-57-7 | sc-295277 sc-295277A | 10 mg 50 mg | $402.00 $1047.00 | ||
L-γ-Carboxyglutamic acid acts as a potent modulator of mGluR-4, characterized by its ability to stabilize receptor conformations and facilitate unique ligand-receptor interactions. This compound influences calcium signaling pathways, enhancing synaptic plasticity through its distinct binding affinity. Its structural features promote specific electrostatic interactions, which can lead to altered receptor activation kinetics, ultimately impacting neuronal excitability and synaptic transmission. | ||||||