RAR Inhibitors
| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
BMS 493 | 215030-90-3 | sc-361124 sc-361124A | 10 mg 50 mg | $459.00 $1428.00 | 7 | |
BMS 493 functions as a selective retinoic acid receptor (RAR) modulator, characterized by its ability to form hydrogen bonds that stabilize receptor-ligand complexes. This compound exhibits a rigid molecular structure, which promotes consistent binding kinetics and enhances specificity for target pathways. Its unique stereochemistry influences the modulation of gene expression, while its hydrophobic regions facilitate interactions with membrane proteins, affecting cellular signaling dynamics. | ||||||
EC 23 | 104561-41-3 | sc-361174 sc-361174A | 5 mg 25 mg | $91.00 $309.00 | 5 | |
EC 23 acts as a retinoic acid receptor (RAR) modulator, distinguished by its capacity to engage in hydrophobic interactions and π-π stacking with receptor domains. This compound demonstrates a selective affinity for specific RAR subtypes, promoting distinct signaling cascades. Its unique steric configuration enhances binding kinetics, allowing for rapid receptor activation. Additionally, EC 23's lipophilic nature contributes to its effective cellular uptake, influencing downstream transcriptional responses. | ||||||
AGN 193109-d7 | 171746-21-7 (unlabeled) | sc-217589 | 1 mg | $453.00 | 1 | |
AGN 193109-d7 acts as a retinoic acid receptor (RAR) modulator, distinguished by its unique conformational flexibility that allows for dynamic interactions with receptor sites. This compound engages in van der Waals forces and hydrophobic interactions, optimizing its affinity for specific RAR subtypes. Its distinct electronic properties enable effective modulation of transcriptional activity, while its solubility characteristics influence cellular uptake and distribution, impacting downstream signaling cascades. | ||||||
AGN 193109 Sodium Salt | 171746-21-7 | sc-210768 sc-210768A | 1 mg 10 mg | $362.00 $2507.00 | 33 | |
AGN 193109 Sodium Salt functions as a retinoic acid receptor (RAR) modulator, characterized by its ability to form stable complexes with receptor proteins through hydrogen bonding and ionic interactions. This compound exhibits a unique ability to alter receptor conformation, enhancing its specificity for various RAR isoforms. Its solubility profile facilitates efficient membrane permeability, influencing its bioavailability and interaction kinetics within cellular environments, thereby affecting gene expression pathways. | ||||||