SR-1B Inhibitors
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Items 11 to 16 of 16 total
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| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
SDZ 21009 | 39731-05-0 | sc-203695 sc-203695A | 10 mg 50 mg | $200.00 $825.00 | ||
SDZ 21009 acts as an SR-1B inhibitor, distinguished by its selective binding to the active site of target proteins, which disrupts their normal function. This compound showcases unique hydrophobic interactions that enhance its affinity, leading to a significant alteration in the protein's structural conformation. Its reaction kinetics indicate a rapid association rate, facilitating effective inhibition. Furthermore, SDZ 21009's unique steric properties influence its interaction dynamics within complex biological systems. | ||||||
Isamoltane hemifumarate | 55050-95-8 | sc-203608 sc-203608A | 10 mg 50 mg | $115.00 $440.00 | ||
Isamoltane hemifumarate functions as an SR-1B inhibitor, characterized by its ability to form stable complexes with target enzymes through specific hydrogen bonding and electrostatic interactions. This compound exhibits a unique conformational flexibility, allowing it to adapt to various binding sites, which enhances its inhibitory efficacy. Its kinetic profile reveals a notable dissociation rate, contributing to prolonged engagement with the target, while its distinct solubility properties facilitate effective distribution in diverse environments. | ||||||
S(−)-Cyanopindolol hemifumarate salt | 874882-72-1 | sc-253460 sc-253460A | 1 mg 5 mg | $197.00 $758.00 | ||
S(-)-Cyanopindolol hemifumarate salt functions as an SR-1B inhibitor, characterized by its ability to form hydrogen bonds with key amino acid side chains, enhancing specificity in target engagement. The compound exhibits a unique conformational flexibility that allows it to adapt to different binding sites, optimizing interaction dynamics. Its distinct electronic properties facilitate charge transfer processes, contributing to its overall reactivity and interaction profile in biological systems. | ||||||
Asenapine maleate | 65576-45-6 | sc-361110 sc-361110A | 10 mg 50 mg | $145.00 $615.00 | ||
Asenapine maleate acts as an SR-1B inhibitor, distinguished by its capacity to engage in intricate π-π stacking interactions with aromatic residues in target proteins. This compound showcases a unique stereochemistry that influences its binding affinity and selectivity. Its reaction kinetics indicate a rapid association phase, followed by a slower dissociation, which supports sustained interaction with the target. Additionally, its amphiphilic nature enhances its solubility in various media, promoting effective molecular interactions. | ||||||
Vortioxetine Hydrobromide | 960203-27-4 | sc-475775 | 5 mg | $220.00 | ||
Vortioxetine Hydrobromide acts as an SR-1B inhibitor, distinguished by its unique ability to modulate serotonin receptor activity through allosteric interactions. The compound's structural features enable it to engage in π-π stacking with aromatic residues, enhancing binding affinity. Its kinetic profile reveals a rapid association and slower dissociation, suggesting prolonged receptor engagement. Additionally, the presence of halogen atoms influences its solubility and molecular interactions, impacting its overall behavior in complex biological environments. | ||||||
GR 127935 hydrochloride | 148642-42-6 | sc-250068 | 10 mg | $209.00 | ||
GR 127935 hydrochloride functions as an SR-1B inhibitor, characterized by its selective binding to receptor sites, which alters downstream signaling pathways. Its unique molecular architecture facilitates hydrogen bonding and hydrophobic interactions, enhancing specificity. The compound exhibits a distinct kinetic behavior, with a notable rate of internalization upon receptor engagement. Furthermore, its ionic nature contributes to its solubility dynamics, influencing interactions within diverse environments. | ||||||