Date published: 2025-11-1

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GR 127935 hydrochloride (CAS 148642-42-6)

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Alternate Names:
N-[4-Methoxy-3-(4-methyl-1-piperazinyl)phenyl]-2'-methyl-4'-(5-methyl-1,2,4-oxadiazol-3-yl)-1,1'-biphenyl-4-carboxamide hydrochloride
Application:
GR 127935 hydrochloride is a selective and potent SR-1B/1D (5-HT1B/1D serotonin receptor) antagonist
CAS Number:
148642-42-6
Purity:
>98%
Molecular Weight:
534.05
Molecular Formula:
C29H31N5O3•HCl
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.

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A selective, potent and orally active 5-HT1B/1D serotonin receptor antagonist.


GR 127935 hydrochloride (CAS 148642-42-6) References

DeVries, P. et al. Br. J. Pharmacol. 118, 85-92, (1996)

Ordering Information

Product NameCatalog #UNITPriceQtyFAVORITES

GR 127935 hydrochloride, 10 mg

sc-250068
10 mg
$209.00