| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
Acamprosate Calcium | 77337-73-6 | sc-210733 | 100 mg | $140.00 | 2 | |
Acamprosate Calcium functions as a modulator of GABAB R1 receptors, exhibiting unique electrostatic interactions that facilitate receptor activation. Its distinct molecular structure allows for specific binding, influencing downstream signaling cascades. The compound's kinetic behavior reveals a slow dissociation rate from the receptor, promoting sustained activity. Additionally, its solubility characteristics enhance its distribution in biological systems, affecting overall receptor engagement and cellular response. | ||||||
(±)-Baclofen | 1134-47-0 | sc-200464 sc-200464A | 1 g 5 g | $56.00 $258.00 | ||
Agonist of GABAB receptors, including GABAB R1, that mimics the effects of GABA, indirectly activating the receptor and modulating neurotransmission. | ||||||
CGP 7930 | 57717-80-3 | sc-203543 sc-203543A | 10 mg 50 mg | $155.00 $625.00 | ||
Positive allosteric modulator of GABAB receptors, enhancing the response to endogenous GABA and indirectly facilitating GABAB R1 activation. | ||||||
Vigabatrin | 60643-86-9 | sc-204382 sc-204382A sc-204382B sc-204382C | 10 mg 50 mg 100 mg 1 g | $125.00 $485.00 $650.00 $1015.00 | 2 | |
GABA transaminase inhibitor that indirectly increases GABA levels in the brain, subsequently enhancing GABAB R1 activation by endogenous GABA. | ||||||
Valproic Acid | 99-66-1 | sc-213144 | 10 g | $87.00 | 9 | |
Enhances GABAergic neurotransmission by inhibiting GABA degradation and indirectly affecting GABAB R1 signaling. | ||||||
Gabapentin | 60142-96-3 | sc-201481 sc-201481A sc-201481B | 20 mg 100 mg 1 g | $53.00 $94.00 $135.00 | 7 | |
Modulates GABAergic signaling, potentially impacting GABAB R1 activity, although its precise mechanism is not fully elucidated. | ||||||
Muscimol | 2763-96-4 | sc-200460 sc-200460A | 5 mg 25 mg | $161.00 $537.00 | 2 | |
Agonist of GABAA receptors, which can indirectly influence GABAB R1 activity through crosstalk between GABA receptor subtypes. | ||||||