Molecular structure of Tyrphostin AG 528, CAS Number: 133550-49-9
Tyrphostin AG 528 (CAS 133550-49-9)
Application:
Tyrphostin AG 528 is an inhibitor of EGFR tyrosine kinase activity
CAS Number:
133550-49-9
Molecular Weight:
306.32
Molecular Formula:
C18H14N2O3
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.
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SDS & Certificate of Analysis
An inhibitor of EGFR protein tyrosine kinase.
Tyrphostin AG 528 (CAS 133550-49-9) References
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- Glycine transporter inhibitors as a novel drug discovery strategy for neuropathic pain. | Dohi, T., et al. 2009. Pharmacol Ther. 123: 54-79. PMID: 19393690
- Modulation of pantothenate kinase 3 activity by small molecules that interact with the substrate/allosteric regulatory domain. | Leonardi, R., et al. 2010. Chem Biol. 17: 892-902. PMID: 20797618
- An image-based, high-throughput screening assay for molecules that induce excess DNA replication in human cancer cells. | Zhu, W., et al. 2011. Mol Cancer Res. 9: 294-310. PMID: 21257818
- Elucidation of crucial structures for a catechol-based inhibitor of plasma hyaluronan-binding protein (factor VII activating protease) autoactivation. | Yamamoto, E., et al. 2011. Biosci Biotechnol Biochem. 75: 2070-2. PMID: 21979097
- Annotated compound data for modulators of detergent-solubilised or lipid-reconstituted respiratory type II NADH dehydrogenase activity obtained by compound library screening. | Dunn, EA., et al. 2016. Data Brief. 6: 275-8. PMID: 26862571
- Investigation of Adsorption Tyrphostin AG528 Anticancer Drug Upon the CNT(6,6-6) Nanotube: A DFT Study. | Sheikhi, M., et al. 2019. Curr Mol Med. 19: 91-104. PMID: 30813875
Inhibitor of:
EGFR, and Tyrosine Kinase.Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
Tyrphostin AG 528, 5 mg | sc-216034 | 5 mg | $42.00 |