Molecular structure of XMD 8-92 (free base), CAS Number: 1234480-50-2
XMD 8-92 (free base) (CAS 1234480-50-2)
See product citations (10)
Application:
XMD 8-92 (free base) is an extremely selective ERK5/BMK1 inhibitor
CAS Number:
1234480-50-2
Molecular Weight:
474.55
Molecular Formula:
C26H30N6O3
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.
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Description
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SDS & Certificate of Analysis
XMD 8-92 is shown to be an extremely selective ERK5/BMK1 inhibitor that presents selectivity over 402 diverse kinases. This compound is shown to be an anti-proliferative agent via inhibition of growth factor-induced activation of cellular BMK1 and reducing of BMK1 activity in in vitro kinase assays.
Inhibitor of:
AIP1, ARID2, DCAMKL2, ERBIN, ERK 3, ERK 5, LOC654106, MAP3K3, Olfr609, Olfr61, PLK4, PRIC285, Rsk, Rsk-4, Ser/Thr Protein Kinase, TRAP230, and UTX.Activator of:
ERK 5, MEF-2C, N-CoR, RYK, and TNIK.Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
XMD 8-92 (free base), 5 mg | sc-364068 | 5 mg | $235.00 | |||
XMD 8-92 (free base), 10 mg | sc-364068A | 10 mg | $340.00 | |||
XMD 8-92 (free base), 100 mg | sc-364068B | 100 mg | $1700.00 | |||
XMD 8-92 (free base), 1 g | sc-364068C | 1 g | $10330.00 |