Hydroxytacrine maleate (CAS 118909-22-1)
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Hydroxytacrine maleate is a compound utilized in the field of chemical research, particularly in studies involving enzyme inhibition. It is structurally related to tacrine, which is known for its inhibitory activity on cholinesterase enzymes. Research involving hydroxytacrine maleate focuses on investigating its potential as an inhibitor for various enzymes, such as acetylcholinesterase and butyrylcholinesterase. These studies help in understanding the structure-activity relationship of cholinesterase inhibitors and the dynamics of enzyme inhibition. The maleate salt form of hydroxytacrine enhances the compound′s solubility in biological media, which is advantageous for in vitro assays. In addition, hydroxytacrine maleate is used to study oxidative stress mechanisms due to its ability to produce reactive oxygen species under certain conditions. This aspect of the compound′s reactivity is of interest in the exploration of the role of oxidative stress in cellular processes. Researchers also examine the interaction of hydroxytacrine maleate with metal ions, which is relevant in the context of metal-mediated neurodegeneration.
Hydroxytacrine maleate (CAS 118909-22-1) References
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Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
Hydroxytacrine maleate, 200 mg | sc-200168 | 200 mg | $69.00 | |||
Hydroxytacrine maleate, 1 g | sc-200168A | 1 g | $264.00 |