(+)-alpha-Methylhistamine dihydrobromide CAS: 75614-93-6
MF: C6H11N3•2HBr
MW: 287
A less active enantiomer of H3 agonist R-(−)-α-methylhistamine.

(+)-α-Methylhistamine dihydrobromide (CAS 75614-93-6)

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Alternate Names: (S)-(+)-α-Methyl-1H-imidazole-4-ethanamine dihydrobromide
Application: (+)-α-Methylhistamine dihydrobromide is a less active enantiomer of H3 agonist R-(−)-α-methylhistamine
CAS Number: 75614-93-6
Molecular Weight: 287
Molecular Formula: C6H11N32HBr
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data (including water content).

(+)-α-Methylhistamine dihydrobromide is the less active enantiomer of histamine H3 receptor agonist R-(-)-α-methylhistamine. 120-fold less potent than R-(-) at H3.


References

Hill (1990) Distribution, properties and functional characteristics of three classes of histamine receptor. Pharmacol.Rev. 42 45.

Physical State :
Solid
Solubility :
Soluble in water (100 mM ).
Storage :
Desiccate at room temperature
Refractive Index :
n20D 1.55 (Predicted)
Optical Activity :
α20/D +3°, c = 1 in water; α25/D +4°, c = 0.8 in water
IC50 :
Histamine H3 receptor: EC5050 = 10 nM (human); Histamine H4 receptor: EC5050 = 12.59 µM (human)
Ki Data :
Histamine H3 receptor: Ki= 50 nM; Histamine H3 receptor: Ki= 63.1 nM (human); Histamine H4 receptor: Ki= 3.98 µM (human)
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
RTECS :
NI3506500
PubChem CID :
45073439
MDL Number :
MFCD00209887
SMILES :
C[[email protected]@H](CC1=CN=CN1)N.Br.Br

Download SDS (MSDS)

Certificate of Analysis

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