Date published: 2026-10-17

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CYP3A 抗体 (D-2): sc-271033

5.0(2)
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说明书
  • CYP3A抗体(D-2)是小鼠单克隆IgG1 κ, 在6篇文献中引用,规格为200 µg/ml
  • 针对氨基酸204-503的抗原,在CYP3A的C-terminus处映射,human来源
  • 推荐用于 mouse, rat 和 human 来源的all CYP3A family members WB, IP, IF 和 ELISA检测
  • 1 BP-HRP">m-IgG1 BP-HRP是CYP3A Antibody (D-2) 适用于 WB 应用。 的首选辅助检测试剂。该试剂现与CYP3A Antibody (D-2) 打包提供(请参阅下面的订购信息)。
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CYP3A基因编码单加氧酶,催化药物代谢和胆固醇、类固醇和其他脂质合成的酶。CYP3A(细胞色素P450,家族3,亚家族A)是人类肝脏中最丰富的p450酶,负责代谢50%以上的所有临床药物。CYP3A成员定位于与药物处置相关的器官,包括肝脏、胃肠道和肾脏。CYP3A簇由四个基因组成:CYP3A43、CYP3A4、CYP3A7和CYP3A5,以及两个假基因:CYP3A5P1和CYP3A5P2。CYP3A簇映射到基因位点7q22.1。

仅限研究使用。不适用于诊断和治疗用途。

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CYP3A 抗体 (D-2) 参考文献:

  1. CYP3A4的功能基因变异。  |  Werk, AN. and Cascorbi, I. 2014. Clin Pharmacol Ther. 96: 340-8. PMID: 24926778
  2. 癌症治疗中CYP3A4介导的药代动力学相互作用。  |  Tian, D. and Hu, Z. 2014. Curr Drug Metab. 15: 808-17. PMID: 25705904
  3. 缺氧下人肝细胞中核受体对CYP3A4的转录调控。  |  Yuan, X., et al. 2020. Drug Metab Rev. 52: 225-234. PMID: 32270716
  4. CRISPR/Cas9编辑的HepG2细胞中CYP3A4和CYP3A5的表达受CYP3A4*1G调控。  |  Yang, W., et al. 2023. Drug Metab Dispos. 51: 492-498. PMID: 36623883
  5. CYP3A4*22可能增加替卡格雷使用者的出血风险。  |  Liedes, H., et al. 2023. Basic Clin Pharmacol Toxicol. 133: 202-207. PMID: 37162098
  6. 强效CYP3A4抑制、CYP3A4诱导和OATP1B1/3抑制对单次口服索托拉西布的药代动力学的影响。  |  Cardona, P., et al. 2024. Clin Pharmacol Drug Dev. 13: 810-818. PMID: 38421129
  7. 总柴胡皂苷对HepaRG细胞中CYP3A4和CYP1A2的影响。  |  Tang, Y., et al. 2024. Exp Ther Med. 27: 217. PMID: 38590569
  8. 卡马西平的药物遗传学:CYP3A4和CYP3A5多态性的系统综述。  |  Riffi, R., et al. 2024. CNS Neurol Disord Drug Targets. 23: 1463-1473. PMID: 38859787
  9. 氯噻隆的CYP3A4介导的代谢活化和细胞毒性。  |  Guo, X., et al. 2024. Chem Res Toxicol. 37: 1104-1112. PMID: 38885202
  10. 奥美拉唑在HepaRG细胞中诱导CYP3A4 mRNA表达,但不诱导CYP3A4蛋白表达。  |  Fujita, Y., et al. 2024. Biol Pharm Bull. 47: 1218-1223. PMID: 38925922

订购信息

产品名称产品编号规格价格数量收藏夹

CYP3A 抗体 (D-2)

sc-271033
200 µg/ml
$322.00

CYP3A (D-2): m-IgG1 BP-HRP 套装

sc-542674
200 µg Ab; 20 µg BP
$361.00

I need to use an antibody to detect the protein in samples of bovine origin. Do you know if sc-271033: CYP3A (D-2) mouse monoclonal antibody will work?

Asked by: AbPolly
Please contact our Technical Service Department and we would be happy to perform sequence analysis and review our data to answer any questions you may have about additional species reactivity.
Answered by: Technical Support
Date published: 2017-03-06
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Rated 5 out of 5 by ET from WB published in rat liver samplesWB published in rat liver samples. -SCBT Publication Review
Date published: 2015-02-02
Rated 5 out of 5 by JM from Good Western blot data obtained in mouseGood Western blot data obtained in mouse liver and human liver tissue extracts. -SCBT QC
Date published: 2014-02-03
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CYP3A抗体 (D-2) is rated 5.0 out of 5 by 2.
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