Molecular structure of Propionylpromazine hydrochloride, CAS Number: 7681-67-6
Propionylpromazine hydrochloride (CAS 7681-67-6)
Alternate Names:
Propiopromazine hydrochloride
Application:
Propionylpromazine hydrochloride is a D2DR inhibitor
CAS Number:
7681-67-6
Purity:
≥93%
Molecular Weight:
376.94
Molecular Formula:
C20H24N2OS•HCl
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.
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SDS & Certificate of Analysis
Propionylpromazine hydrochloride is a dopamine receptor antagonist. It acts by blocking the dopamine receptors in the central nervous system. This blockade results in a decrease in the effects of dopamine, leading to sedative and antiemetic effects. Propionylpromazine hydrochloride may possess antipsychotic properties due to its ability to modulate dopamine neurotransmission. Its mechanism of action involves inhibiting the release of dopamine and altering the sensitivity of dopamine receptors in the brain. Propionylpromazine Hydrochloride also exhibits anticholinergic and alpha-adrenergic blocking properties, contributing to its pharmacological effects.
Propionylpromazine hydrochloride (CAS 7681-67-6) References
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- Metabolism and pharmacokinetic studies of propionylpromazine in horses. | Park, J., et al. 1989. J Chromatogr. 489: 313-21. PMID: 2753955
- Effect of phenothiazine compounds on the secondary structure and fibrillogenesis of poly-l-lysine. | Cieślik-Boczula, K. 2019. Spectrochim Acta A Mol Biomol Spectrosc. 216: 15-24. PMID: 30870786
- Screening for modulators of neural network activity in 3D human iPSC-derived cortical spheroids. | Woodruff, G., et al. 2020. PLoS One. 15: e0240991. PMID: 33091047
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Inhibitor of:
D2DR.Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
Propionylpromazine hydrochloride, 100 mg | sc-250790 | 100 mg | $84.00 |