| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
KT 5720 | 108068-98-0 | sc-3538 sc-3538A sc-3538B | 50 µg 100 µg 500 µg | $138.00 $220.00 $972.00 | 47 | |
KT 5720, functioning as a potent PHK, uniquely interacts with protein kinases, particularly influencing the phosphorylation state of serine and threonine residues. Its structural conformation facilitates selective inhibition, altering kinase activity and downstream signaling pathways. The compound's kinetic properties allow for rapid binding and dissociation, enhancing its regulatory potential in cellular processes. Furthermore, its solubility in diverse solvents supports versatile interactions within complex biochemical systems. | ||||||
Bisindolylmaleimide I (GF 109203X) | 133052-90-1 | sc-24003A sc-24003 | 1 mg 5 mg | $105.00 $242.00 | 36 | |
Bisindolylmaleimide I (GF 109203X) acts as a selective protein kinase inhibitor, exhibiting a unique ability to stabilize the inactive conformation of kinases. This compound engages in specific hydrogen bonding and hydrophobic interactions, which modulate enzyme activity and influence cellular signaling cascades. Its distinct molecular architecture allows for targeted inhibition, while its favorable solubility profile enhances its compatibility with various biochemical environments, promoting effective engagement with multiple kinase targets. | ||||||
K-252a | 99533-80-9 | sc-200517 sc-200517B sc-200517A | 100 µg 500 µg 1 mg | $129.00 $214.00 $498.00 | 19 | |
K-252a is a potent inhibitor of protein kinases, characterized by its ability to disrupt ATP binding through unique interactions with the enzyme's active site. This compound exhibits a distinctive binding affinity, facilitating conformational changes that hinder kinase activation. Its structural features promote specific van der Waals and electrostatic interactions, enhancing selectivity. Additionally, K-252a's solubility in diverse solvents allows for versatile applications in biochemical assays, making it a valuable tool for studying kinase dynamics. | ||||||