Molecular structure of Ziprasidone hydrochloride monohydrate, CAS Number: 138982-67-9
Ziprasidone hydrochloride monohydrate (CAS 138982-67-9)
Application:
Ziprasidone hydrochloride monohydrate is an SR-2A and D2DR inhibitor
CAS Number:
138982-67-9
Purity:
≥98%
Molecular Weight:
467.4
Molecular Formula:
C21H21ClN4OS•HCl•H2O
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.
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Description
Technical Information
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SDS & Certificate of Analysis
Ziprasidone hydrochloride monohydrate is an atypical antipsychotic that displays combined SR-2A and D2DR inhibition. Ziprasidone displays high affinity at SR-2A receptors with a SR-2A/D2DR affinity ratio greater than any other clinically available atypical antipsychotics (pKi values are 9.38, 8.88, 8.69, 8.47, 8.32, 8.14, 7.98, 7.49, 7.33 and 6.28 for SR-2A, 5-HT2C, 5-HT1D, 5-HT1A, D2DR, D3, α1, D4, H1 and D1 receptors respectively).
Ziprasidone hydrochloride monohydrate (CAS 138982-67-9) References
Seeger et al (1995) Ziprasidone (CP-88,059): a new antipsychotic with combined dopamine and serotonin receptor antagonist activity. J.Pharmacol.Exp.Ther. 275 101. Schmidt et al (2001) Ziprasidone: a novel antipsychotic agent with a unique human receptor binding profile. Eur.J.Pharmacol. 425 197. Fell et al (2005) Investigation into the effects of the novel antipsychotic ziprasidone on weight gain and reproductive function in female rats. Behav.Brain Res. 160 338.Inhibitor of:
D2DR, SR-1B, SR-1D, and SR-2A.Activator of:
SR-1A.Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
Ziprasidone hydrochloride monohydrate, 10 mg | sc-204419 | 10 mg | $125.00 | |||
Ziprasidone hydrochloride monohydrate, 50 mg | sc-204419A | 50 mg | $525.00 |