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Zatebradine hydrochloride is a bradycardic agent that creates use-dependent inhibition of hyperpolarization-activated current (If) in sinoatrial node cells (EC50 = 480 nM) and Purkinje fibres. Displays negative chronotropic activity in isolated guinea pig atria (EC50 of 13.4μM).
Ordering Information
Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
Zatebradine hydrochloride, 10 mg | sc-500908 | 10 mg | $206.00 | |||
Zatebradine hydrochloride, 50 mg | sc-500908A | 50 mg | $760.00 |