Xylometazoline hydrochloride, α-adrenoceptor agonist; imidazoline binding site ligand. Xylometazoline hydrochloride is an activator of α1A-AR, α1B-AR, α1D-AR, α2A-AR, α2B-AR and α2C-AR.
Sakuta, H., and Okamoto, K., Inhibition by imidazoline and imidazolidine derivatives of glibenclamide-sensitive K+ currents in Xenopus oocytes. Eur. J. Pharmacol. 259, 223-231, (1994) Bognar, I.T., et al., å-adrenoceptor mediated facilitation of acetylcholine release in the rat perfused heart. J. Pharmacol. Exp. Ther. 254, 702, (1990)
Soluble in ethanol (100 mg/ml), and DMSO (27 mg/ml at 25° C).
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