TPMPA (CAS 182485-36-5)
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TPMPA is a competitive, selective GABAC antagonist with minimal effects on GABAA and GABAB receptors (Kb values are 2.1 muM (antagonist), 320 muM (antagonist) and EC50 ~ 500 muM (weak agonist) respectively). Shows 8-fold selectivity for human recombinant rho 1 receptors. TPMPA, a synthetic molecule, has recently captured the attention of the scientific community owing to its potential applications across diverse research domains. The compound, also known as 4-Methyl-2-Phenyl-2-Propanol, shares a structural resemblance with the neurotransmitter dopamine and belongs to the aniline derivative class. Its significance lies in its capacity to engage with dopamine receptors and influence the brain′s response to dopamine.
TPMPA (CAS 182485-36-5) References
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Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
TPMPA, 10 mg | sc-204352 | 10 mg | $307.00 | |||
TPMPA, 50 mg | sc-204352A | 50 mg | $864.00 |