Molecular structure of Tianeptine, CAS Number: 66981-73-5
Tianeptine (CAS 66981-73-5)
Application:
Tianeptine is a selective facilitator of serotonin uptake
CAS Number:
66981-73-5
Molecular Weight:
436.95
Molecular Formula:
C21H25ClN2O4S
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.
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SDS & Certificate of Analysis
Tianeptine, a tricyclic compound, is a selective facilitator of 5-HT (serotonin sc-201146) uptake in vitro and in vivo. Additionally, Tianeptine is reported to act as a selective inhibitor of dopamine uptake and is similar to amineptine. Tianeptine does not have a noted effect on monoamine uptake. In a study utilizing purified synaptosomes from rat brain, Tianeptine was reported to enhance serotonin uptake in selective brain regions. Purified synaptosomes were obtained from rats and incubated with tritium-labeled 5-H and Tianeptine in vitro. The synaptosomes were then analyzed for uptake and release of 5-HT via a liquid scintillation counter.
Tianeptine (CAS 66981-73-5) References
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Inhibitor of:
MDMA, Shank2, and Slc6a16.Activator of:
1700016H13Rik, Arc, Cerebellin 3, Cerebellin 4, dendrin, EAAT4, GRINA, Homer-2, Homer-3, IMP-1, Latrophilin-3, M6A, neugrin, Neuroplastin, oligophrenin-1, PSD-95, SAPAP2, SHISA9, VGLUT1, and VMAT 2.Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
Tianeptine, 10 mg | sc-213044 | 10 mg | $250.00 | |||
Tianeptine, 50 mg | sc-213044A | 50 mg | $422.00 |