Tetradecyl Phosphonate is a pan-antagonist of EDG-2, EDG-4, and EDG-7 (EDG-2, EDG-4, and EDG-7 receptors) with IC50 values for inhibition of EDG-induced calcium mobilization of 10 μM, 5.5 μM, and 3.1 μM, respectively. Tetradecyl Phosphonate is an inhibitor of Autotaxin.
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