Molecular structure of TAK-960, CAS Number: 1137868-52-0
TAK-960 (CAS 1137868-52-0)
See product citations (1)
Application:
TAK-960 is a Plk inhibitor
CAS Number:
1137868-52-0
Purity:
>98%
Molecular Weight:
561.6
Molecular Formula:
C27H34F3N7O3
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.
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Description
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SDS & Certificate of Analysis
TAK-960 has shown activity in several tumor cell lines including those that express multi-drug resistant protein 1 (MDR1). Consistent with PLK1 inhibition, TAK-960 treatment gives rise to accumulation of G2/M cells, aberrant "polo" mitosis morphology, and increases phosphorylation of histone H3 (pHH3). TAK-960 inhibits proliferation of multiple cancer cell lines, with mean EC50 values ranging from 8.4 to 46.9 nM. TAK-960 is an inhibitor of Plk.
Inhibitor of:
Plk.Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
TAK-960, 5 mg | sc-364631 | 5 mg | $310.00 | |||
TAK-960, 10 mg | sc-364631A | 10 mg | $653.00 |