Molecular structure of (S)-4C3H-PG, CAS Number: 85148-82-9
(S)-4C3H-PG (CAS 85148-82-9)
Application:
(S)-4C3H-PG is an agonist for group II mGluRs and competitive antagonist for group I mGluR
CAS Number:
85148-82-9
Molecular Weight:
211.17
Molecular Formula:
C9H9NO5
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.
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SDS & Certificate of Analysis
(S)-4C3H-PG is an agonist for group II mGluR (mGluR-2 and mGluR-3). (S)-4C3H-PG also acts as a competitive antagonist for group I mGluR-1 and exhibits mixed effects at mGluR-5. (S)-4C3H-PG is an inhibitor of mGluR-1a.
(S)-4C3H-PG (CAS 85148-82-9) References
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- Metabotropic receptors in excitotoxicity: (S)-4-carboxy-3-hydroxyphenylglycine ((S)-4C3HPG) protects against rat striatal quinolinic acid lesions. | Orlando, LR., et al. 1995. Neurosci Lett. 202: 109-12. PMID: 8787843
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- (S)-4-carboxy-3-hydroxyphenylglycine activates phosphatidyl inositol linked metabotropic glutamate receptors in different brain regions of the neonatal rat. | Sacaan, AI., et al. 1998. Neurochem Int. 32: 77-85. PMID: 9460705
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Inhibitor of:
mGluR-1a, and mGluR-5.Activator of:
mGluR-2, mGluR-3, mGluR-5, and mGLuR-8.Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
(S)-4C3H-PG, 1 mg | sc-203249 | 1 mg | $30.00 | |||
(S)-4C3H-PG, 5 mg | sc-203249A | 5 mg | $123.00 |