RS-127445 (CAS 199864-87-4)
Alternate Names:
4-(4-fluoro-1-naphthalenyl)-6-(1-methylethyl)-2-pyrimidinamine
Application:
RS-127445 is a 5-HT2B receptor antagonist with modest activity against other 5-HT receptors
CAS Number:
199864-87-4
Molecular Weight:
281.3
Molecular Formula:
C17H16FN3
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.
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Description
Technical Information
Safety Information
SDS & Certificate of Analysis
RS-127445 is a high affinity 5-HT2B receptor antagonist with a pIC50 of 10.4. The pKi of RS-127445 for the 5-HT2B receptor is 9.5. RS-127445 has 1000 fold selectivity over the human recombinant 5-HT2A, 5-HT2C, 5-HT5, 5-HT6 and 5-HT7 receptors.
Inhibitor of:
Serotonin.Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
RS-127445, 5 mg | sc-364604 | 5 mg | $105.00 | |||
RS-127445, 50 mg | sc-364604A | 50 mg | $700.00 |