Ritanserin is a potent and long-acting SR-2A (5-HT2 receptor) antagonist (Ki = 0.39 nM).
Janssen (1985) Pharmacology of potent and selective S2-serotonergic antagonists. J.Cardiovasc.Pharmacol. 7 S2. Leysen et al (1985) Receptor-binding properties in vitro and in vivo of ritanserin. Mol.Pharmacol. 27 600. Watanabe et al (1992) Syntheses and 5
Soluble in water (1.3 mg/ml), ethanol (25 mM), DMSO (100 mM), and methanol (>10 mg/ml). Insoluble in dilute aqueous base.
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GarciaGarcia-Pedraza el al. (PubMed ID 25854421) used Ritanserin to inactivate 5-HT and prevent vasoconstriction to study 5-HT1D activation by nitric oxide. -SCBT Publication Review
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