Date published: 2025-9-5

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PTP CD45 Inhibitor 抑制剂 (CAS 345630-40-2)

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备用名:
Protein Tyrosine Phosphatase CD45 Inhibitor; N-(9,10-dihydro-9,10-dioxo-2-phenanthrenyl)-2,2-dimethyl-propanamide
应用:
PTP CD45 Inhibitor 是一种具有细胞渗透性的 CD45 强效可逆抑制剂
CAS号码:
345630-40-2
纯度:
≥97%
分子量:
307.34
分子式:
C19H17NO3
仅供科研使用。不可用于诊断或治疗。
* 参考分析证明 大量特定数据 (包括水 含量).

快捷链接

PTP CD45 Inhibitor是一种细胞可渗透的、强效的、选择性的、竞争性的、可逆的CD45抑制剂(分别使用pNPP或磷酸化Ick505肽作为底物,IC50 = 200 nM或3.8 μM)。PTP CD45 Inhibitor无法有效抑制PTPIB(使用磷酸化Ick505肽作为底物,IC50


PTP CD45 Inhibitor 抑制剂 (CAS 345630-40-2) 参考文献

  1. 蛋白酪氨酸磷酸酶 CD45 的强效可逆抑制剂。  |  Urbanek, RA., et al. 2001. J Med Chem. 44: 1777-93. PMID: 11356112
  2. GM1控制的酪氨酸激酶Lck横向分离使T细胞易受细胞衍生的galectin-1诱导的细胞凋亡影响。  |  Novák, J., et al. 2014. Mol Immunol. 57: 302-9. PMID: 24231767
  3. 分化簇 45 的激活在白细胞介素-10 依赖性肿瘤相关树突状细胞分化过程中至关重要。  |  Cheng, DE., et al. 2014. Oncol Lett. 8: 620-626. PMID: 25013476
  4. T 辅助信号通过上调 CD45 磷酸酶的活性,恢复自反应性过敏 B 细胞的 B 细胞受体信号转导。  |  Szodoray, P., et al. 2016. J Allergy Clin Immunol. 138: 839-851.e8. PMID: 27056269
  5. 利用基因编码的 NAD+/NADH 传感器对活细胞中的线粒体代谢状态进行实时和高通量分析。  |  Zhao, Y. and Yang, Y. 2016. Free Radic Biol Med. 100: 43-52. PMID: 27261194
  6. 利用基因编码荧光传感器实现烟碱腺嘌呤二核苷酸氧化还原平衡的可视化。  |  Zhao, Y., et al. 2018. Antioxid Redox Signal. 28: 213-229. PMID: 28648094
  7. 真菌Clitocybe nebularis凝集素与不同的细胞表面糖蛋白受体结合,选择性地诱导Jurkat细胞死亡。  |  Perišić Nanut, M., et al. 2022. FASEB J. 36: e22215. PMID: 35224765
  8. T 辅助细胞通过 galectin-1 和 CD43 调节 CD45 磷酸酶的活性,从而控制慢性淋巴细胞白血病的增殖。  |  Imbery, JF., et al. 2022. Br J Haematol. 198: 556-573. PMID: 35655388

订购信息

产品名称产品编号规格价格数量收藏夹

PTP CD45 Inhibitor, 1 mg

sc-222223A
1 mg
$102.00

PTP CD45 Inhibitor, 5 mg

sc-222223
5 mg
$300.00

你好 请问此抑制剂可以通过侧脑室注射达到抑制脑内cd45的作用么

Asked by: xibp
感谢您的提问。如果您能直接拨打(+86) 021-60936350,或者发邮件到我们亚洲服务部的邮箱asia@scbio.cn我们就这个问题和其他相关问题进行更多的互动讨论,那将会很有帮助。 Thank you for your question.It would be helpful if you could call us directly at (+86) 021-60936350 or email our Asia Service department at asia@scbio.cn for more interactive discussions on this and other related issues.
Answered by: Zhanglong
Date published: 2024-05-20

Please provide a detailed protocol of the PTP CD 45 inhibitor for cell culture study. want to use on mesenchymal stem cells from mouse bone marrow

Asked by: Madhurima
Thank you for your question. It would be helpful if you could call 800-457-3801, allowing for a more interactive discussion of this and other related questions.
Answered by: Technical Service
Date published: 2022-09-06
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Rated 5 out of 5 by from Great PurchaseExcellent purchase. Quality is very high. I will order again
Date published: 2021-08-06
Rated 5 out of 5 by from PTP CD45 Inhibitor was found to inhibit thePTP CD45 Inhibitor was found to inhibit the action of lambda protein phosphatase. This was demonstrated by IF showing nuclear localization and increase in signal of phosphorylated NFkB p50 in the treated NIH/3T3 cells. -SCBT QC
Date published: 2015-02-16
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PTP CD45 Inhibitor 抑制剂 is rated 5.0 out of 5 by 2.
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