(±)-5′-Chloro-5′-deoxy-ENBA is a highly selective Adenosine A1-R agonist (Ki values are 0.51, 1290, 1340 and 2740 at Adenosine A1-R, Adenosine A3-R, Adenosine A2A-R and Adenosine A2B-R, respectively). (±)-5′-Chloro-5′-deoxy-ENBA is also an antinociceptive.
1. Trivedi, B.K, et al. 1989. J. Med. Chem. 32: 8-11. PMID: 2909748 2. Franchetti, P., et al. 2009. J. Med. Chem. 52: 2393-2406. PMID: 19317449
To place an order using RMB or to ship to mainland China, please visit www.scbio.cn