Date published: 2025-10-15

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Naltriben methanesulfonate (CAS 111555-58-9)

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Alternate Names:
NTB
Application:
Naltriben methanesulfonate is a highly selective δ2 opioid receptor (DOR) antagonist
CAS Number:
111555-58-9
Molecular Weight:
511.59 (anhydrous basis)
Molecular Formula:
C26H25NO4•CH4O3S•xH2O
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.

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Naltriben methanesulfonate is a highly selective DOR (delta2 opioid receptor) antagonist. Ligand binding assays show biphasic binding of the antagonist to the single receptor type. Naltriben methanesulfonate is a highly effective and specific inhibitor of Bruton′s tyrosine kinase (BTK), which effectively hinders the activation of B-cells. This compound serves as a valuable research tool for investigating the role of BTK in various cellular processes, including the examination of peptides and proteins that interact with this kinase. Additionally, it exhibits inhibitory properties against protein interactions involving the receptor for advanced glycation endproducts (RAGE).


Naltriben methanesulfonate (CAS 111555-58-9) References

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  8. Function and regulation of TRPM7, as well as intracellular magnesium content, are altered in cells expressing ΔF508-CFTR and G551D-CFTR.  |  Huguet, F., et al. 2016. Cell Mol Life Sci. 73: 3351-73. PMID: 26874684
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Ordering Information

Product NameCatalog #UNITPriceQtyFAVORITES

Naltriben methanesulfonate, 1 mg

sc-301456A
1 mg
$122.00

Naltriben methanesulfonate, 5 mg

sc-301456
5 mg
$195.00

Naltriben methanesulfonate, 25 mg

sc-301456B
25 mg
$632.00