Molecular structure of N-Cyclobutanecarbonyl-2-phenyltryptamine
N-Cyclobutanecarbonyl-2-phenyltryptamine
Application:
N-Cyclobutanecarbonyl-2-phenyltryptamine is a MEL-1 (melatonin receptor) antagonist
Molecular Weight:
318.41
Molecular Formula:
C21H22N2O
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.
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Description
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SDS & Certificate of Analysis
N-Cyclobutanecarbonyl-2-phenyltryptamine is a melatonin receptor antagonist. It is more potent compared to Luzindole (sc-202700) in the Xenopus melanophore assay.
N-Cyclobutanecarbonyl-2-phenyltryptamine References
- Mapping the melatonin receptor. 3. Design and synthesis of melatonin agonists and antagonists derived from 2-phenyltryptamines. | Garratt, PJ., et al. 1995. J Med Chem. 38: 1132-9. PMID: 7707316
- Radioligand binding affinity and biological activity of the enantiomers of a chiral melatonin analogue. | Sugden, D., et al. 1995. Eur J Pharmacol. 287: 239-43. PMID: 8991796
- Mapping the melatonin receptor. 5. Melatonin agonists and antagonists derived from tetrahydrocyclopent[b]indoles, tetrahydrocarbazoles and hexahydrocyclohept[b]indoles. | Davies, DJ., et al. 1998. J Med Chem. 41: 451-67. PMID: 9484496
Inhibitor of:
MEL-1.Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
N-Cyclobutanecarbonyl-2-phenyltryptamine, 1 mg | sc-221998 | 1 mg | $41.00 | |||
N-Cyclobutanecarbonyl-2-phenyltryptamine, 5 mg | sc-221998A | 5 mg | $123.00 |