Molecular structure of MSK-195, CAS Number: 289902-82-5
MSK-195 (CAS 289902-82-5)
See product citations (1)
Alternate Names:
N-[2-(3,4-Dimethylbenzyl)-3-(pivalyloxy)propyl]-2-[4-(2-aminoethoxy)-3-methoxyphenyl]acetamide
Application:
MSK-195 is a potentially useful biochemical with RTX binding affinity and agonism
CAS Number:
289902-82-5
Purity:
≥98%
Molecular Weight:
484.6
Molecular Formula:
C28H40N2O5
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.
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SDS & Certificate of Analysis
MSK-195 is a potent analgesic with EC50 = 0.96 μg/kg in the acetic acid-induced writhing test. RTX binding affinity (Ki = 603 nM), agonism (calcium influx; EC50 = 240 nM).
MSK-195 (CAS 289902-82-5) References
Phenolic modification as an approach to improve the pharmacology of the 3-acyloxy-2-benzylpropyl homovanillic amides and thioureas, a promising class of vanilloid receptor agonists and analgesics: J. Lee, et al.; Bioorg. Med. Chem. 10, 1171 (2002)Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
MSK-195, 1 mg | sc-202712 | 1 mg | $77.00 | |||
MSK-195, 5 mg | sc-202712A | 5 mg | $287.00 |