Molecular structure of (−)-Bicuculline methochloride, CAS Number: 53552-05-9
(−)-Bicuculline methochloride (CAS 53552-05-9)
Application:
(−)-Bicuculline methochloride is a water-soluble GABAA antagonist
CAS Number:
53552-05-9
Molecular Weight:
417.84
Molecular Formula:
C21H20ClNO6
Supplemental Information:
This is classified as a Dangerous Good for transport and may be subject to additional shipping charges.
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.
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SDS & Certificate of Analysis
(−)-Bicuculline methochloride is a methochloride salt of (+)-bicuculline. This compound is a water-soluble GABA Receptor (GABAA) antagonist. (−)-Bicuculline methochloride is more stable than bicuculline, and non-GABA receptor-mediated actions are reported.
(−)-Bicuculline methochloride (CAS 53552-05-9) References
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- The actions of cimetidine, mepyramine, indomethacin and aprotinin (Trasylol) on the inflammatory response in adjuvant rats [proceedings]. | Al-Haboubi, HA. and Zeitlin, IJ. 1979. Br J Pharmacol. 67: 446P-447P. PMID: 315249
- The quantal size at retinogeniculate synapses determined from spontaneous and evoked EPSCs in guinea-pig thalamic slices. | Paulsen, O. and Heggelund, P. 1994. J Physiol. 480 (Pt 3): 505-11. PMID: 7869264
- Quantal properties of spontaneous EPSCs in neurones of the guinea-pig dorsal lateral geniculate nucleus. | Paulsen, O. and Heggelund, P. 1996. J Physiol. 496 (Pt 3): 759-72. PMID: 8930842
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Inhibitor of:
GABA Receptor.Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
(−)-Bicuculline methochloride, 10 mg | sc-203528 | 10 mg | $138.00 | |||
(−)-Bicuculline methochloride, 50 mg | sc-203528A | 50 mg | $635.00 | |||
(−)-Bicuculline methochloride, 500 mg | sc-203528B | 500 mg | $5200.00 |