Molecular structure of LU AA33810, CAS Number: 304008-29-5
LU AA33810 (CAS 304008-29-5)
Alternate Names:
N-[[trans-4-[(4,5-Dihydro[1]benzothiepino[5,4-d]thiazol-2-yl)amino]cyclohexyl]methyl]methanesulfonamide
Application:
LU AA33810 is a potent NPY5-R antagonist
CAS Number:
304008-29-5
Molecular Weight:
423.62
Molecular Formula:
C19H25N3O2S3
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
Available in US only.
Available in US only.
* Refer to Certificate of Analysis for lot specific data.
QUICK LINKS
Ordering Information
Description
Technical Information
Safety Information
SDS & Certificate of Analysis
A potent neuropeptide Y (NPY) Y5 receptor antagonist. Displays ≥ 3300-fold affinity for Y5 over Y1, Y2 and Y4 receptors. Also binds human 5-HT2B and 5-HT1A receptors (Ki values are 247 and 478 nM respectively). Exerts anxiolytic- and antidepressant-like effects in rat models of stress sensitivity.
LU AA33810 (CAS 304008-29-5) References
Walker et al (2009) The novel neuropeptide Y Y5 receptor antagonist Lu AA33810 [N-[[trans-4-[(4,5-dihydro[1]benzothiepino[5,4-d]thiazol-2-yl)amino]cyclohexyl]methyl]-methanesulfonamide] exerts anxiolytic- and antidepressant-like effects in rat models of stress anxiety. J.Pharmacol.Exp.Ther. 328 900.Inhibitor of:
NPY Receptor, and NPY5-R.Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
LU AA33810, 10 mg | sc-295367 | 10 mg | $169.00 | |||
| US: Only available in the US | ||||||
LU AA33810, 50 mg | sc-295367A | 50 mg | $638.00 | |||
| US: Only available in the US | ||||||