Molecular structure of L-803,087 trifluoroacetate, CAS Number: 217480-26-7
L-803,087 trifluoroacetate (CAS 217480-26-7)
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Alternate Names:
N2-[4-(5,7-Difluoro-2-phenyl-1H-indol-3-yl)-1-oxobutyl]-L-arginine methyl ester trifluoroacetate
Application:
L-803,087 trifluoroacetate is a potent and selective sst4 agonist
CAS Number:
217480-26-7
Purity:
≥97%
Molecular Weight:
599.56
Molecular Formula:
C25H29F2N5O3•CF3CO2H
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
Available in US only.
Available in US only.
* Refer to Certificate of Analysis for lot specific data.
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Description
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SDS & Certificate of Analysis
Potent and selective sst4 agonist Potent and selective somatostatin sst4 receptor agonist. Ki values are 0.7, 199, 4720, 1280 and 3880 nM for cloned human sst4, sst1, sst2, sst3 and sst5 receptors respectively. Facilitates AMPA-mediated hippocampal synaptic responses in vitro.
L-803,087 trifluoroacetate (CAS 217480-26-7) References
- Somatostatin inhibits colon cancer cell growth through cyclooxygenase-2 downregulation. | Colucci, R., et al. 2008. Br J Pharmacol. 155: 198-209. PMID: 18587421
- Modulation of voltage-gated ion channels in rat retinal ganglion cells mediated by somatostatin receptor subtype 4. | Farrell, SR., et al. 2010. J Neurophysiol. 104: 1347-54. PMID: 20573967
- Parallel Inhibition of Dopamine Amacrine Cells and Intrinsically Photosensitive Retinal Ganglion Cells in a Non-Image-Forming Visual Circuit of the Mouse Retina. | Vuong, HE., et al. 2015. J Neurosci. 35: 15955-70. PMID: 26631476
Activator of:
SSTR4, and SSTR5.Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
L-803,087 trifluoroacetate, 10 mg | sc-203619 | 10 mg | $320.00 | |||
| US: Only available in the US | ||||||